リルメニジン

MSDS Information

• Oxaminozoline

リルメニジン 化学特性,用途語,生産方法

• 効能

  血圧降下薬, α2アドレナリン受容体作動薬

• 説明

  Rilmenidine is a new antihypertensive agent with a selective alphaz-agonist/antagonist profile, reportedly useful in the management of mild to moderate hypertension. Its fmt-line indication is possible because of the clear dissociation of its antihypertensive activity from other neurophannacological effects.

• 化学的特性

  water soluble

• 使用

  I1-imidazoline binding site ligand and a2-adrenoceptor agonist, exhibits higher I1 vs. a2 selectivity than clonidine

• 生物活性

  I 1 -imidazoline binding site selective ligand and α 2 -adrenoceptor agonist. Possesses greater I 1 vs α 2 selectivity than the prototypical compound, clonidine.

• 代謝経路

  In short-term rat hepatocyte cultures, oxaminozoline is metabolized and its four metabolites resulting from oxidation or hydrolysis are identified, three of which are identical to those reported in vivo. The presence of an additional minor metabolite in culture may be due to the higher metabolic rate of oxaminozoline in this model system.

リルメニジン 上流と下流の製品情報

リルメニジン 生産企業

Global(130)Suppliers

54187-04-1, リルメニジン キーワード