网站主页 化工产品目录 原料药
抗肿瘤药
替尼类抗肿瘤药
Hexanedioic acid, compd. with (6R)-7-[(3,4-difluorophenyl)methyl]-6,7-dihydro-6-(methoxymethyl)-2-[5-methyl-2-[(1-methyl-1H-pyrazol-5-yl)amino]-4-pyrimidinyl]imidazo[1,2-a]pyrazin-8(5H)-one (1:2)
Hexanedioic acid, compd. with (6R)-7-[(3,4-difluorophenyl)methyl]-6,7-dihydro-6-(methoxymethyl)-2-[5-methyl-2-[(1-methyl-1H-pyrazol-5-yl)amino]-4-pyrimidinyl]imidazo[1,2-a]pyrazin-8(5H)-one (1:2)
Hexanedioic acid, compd. with (6R)-7-[(3,4-difluorophenyl)methyl]-6,7-dihydro-6-(methoxymethyl)-2-[5-methyl-2-[(1-methyl-1H-pyrazol-5-yl)amino]-4-pyrimidinyl]imidazo[1,2-a]pyrazin-8(5H)-one (1:2)
英文名称:Hexanedioic acid, compd. with (6R)-7-[(3,4-difluorophenyl)methyl]-6,7-dihydro-6-(methoxymethyl)-2-[5-methyl-2-[(1-methyl-1H-pyrazol-5-yl)amino]-4-pyrimidinyl]imidazo[1,2-a]pyrazin-8(5H)-one (1:2)
CAS号:2097416-93-6
分子式:C24H24F2N8O2.1/2C6H10O4
分子量:1135.14
EINECS号:
Mol文件:2097416-93-6.mol
Hexanedioic acid, compd. with (6R)-7-[(3,4-difluorophenyl)methyl]-6,7-dihydro-6-(methoxymethyl)-2-[5-methyl-2-[(1-methyl-1H-pyrazol-5-yl)amino]-4-pyrimidinyl]imidazo[1,2-a]pyrazin-8(5H)-one (1:2) 用途与合成方法
Tizaterkib hexanedioic acid (example 18) 是一种有效的选择性 ERK2 抑制剂,IC50 为 0.6 nM。