1881233-39-1
1881233-39-1 性质
密度 | 1.367±0.06 g/cm3(Predicted) |
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储存条件 | Store at -20°C |
溶解度 | 二甲基亚砜:≥30 mg/ml(63.08mM) |
形态 | 固体 |
酸度系数(pKa) | 9.06±0.10(Predicted) |
颜色 | 白色至米白色 |
1881233-39-1 用途与合成方法
PI4KIIIβ 3.6 nM (IC 50 ) |
PI4KIIIα 3 μM (IC 50 ) |
PI3Kδ 720 nM (IC 50 ) |
PI3KC2γ 1 μM (IC 50 ) |
PI3Kα 10 μM (IC 50 ) |
PI3Kγ 20 μM (IC 50 ) |
PI4KIIIbeta-IN-10 (Compound 10) is a potent PI4KIIIβ inhibitor with very minor off-target inhibition of PI4KIIIβ related lipid kinases. PI4KIIIbeta-IN-10 shows weak inhibition of PI3KC2γ (IC 50 ~1 µM), PI3Kα (~10 µM), and PI4KIIIα (~3 µM), and <20% inhibition at concentrations up to 20 µM for PI4K2α, PI4K2β, and PI3Kβ.
1881233-39-1 价格(试剂级)
更新日期 | 产品编号 | 产品名称 | CAS号 | 包装 | 价格 |
---|---|---|---|---|---|
2024-11-08 | HY-100198 | 1881233-39-1 | 1881233-39-1 | 1mg | 1300 |
2024-11-08 | HY-100198 | 1881233-39-1 | 1881233-39-1 | 5mg | 2900 |