RepSox

Product Description

RepSox is a potent and selective inhibitor of the TGFβR-1/ALK5 with IC50 of 23 nM and 4 nM for ATP binding to ALK5 and ALK5 autophosphorylation, respectively.

Target

TGFβR1(ALK5)

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IC50 Value

4nM

Diseases and Conditions

Immunology

体外

体内

分子量

287.32

储存条件

分子式

C₁₇H₁₃N₅

CAS:

446859-33-2

备注

For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.

溶解度

体外

Ethanol

DMSO

57mg/ml(198.39 mM)

Water

<1mg/ml

体内

* <1 mg/ml refers to the product slightly soluble or insoluble

浓度溶解体积质量

1mg

5mg

10mg

1mM

3.4804mL

17.4022mL