Triptorelin Acetate

Chemical Name:Triptorelin Acetate

Synonyms:Decapeptyl, Gonapeptyl, Triptorelinum

CAS Number:57773-63-4

Molecular Formula:C₆₄H₈₂N₁₈O₁₃ · C₂H₄O₂

Molecular Weight:1311.46 g/mol (free base) + 60.05 g/mol (acetic acid) = 1371.51 g/mol (total)

Appearance:White to off-white powder

Solubility: Soluble in water, slightly soluble in ethanol

Storage Conditions :Store at 2-8°C, protected from light and moisture

Stability:Stable under recommended storage conditions

Pharmacological Class:Gonadotropin-releasing hormone (GnRH) agonist

Therapeutic Use:Treatment of prostate cancer, endometriosis, and central precocious puberty

Mechanism of Action:Initially stimulates, then suppresses the release of gonadotropins (LH and FSH)

Half-life:Approximately 2-4 hours (after subcutaneous or intramuscular injection)

Route of Administration:Subcutaneous or intramuscular injection

Triptorelin Acetate is a synthetic decapeptide analog of gonadotropin-releasing hormone (GnRH). It acts as a potent agonist of GnRH receptors, initially stimulating the release of luteinizing hormone (LH) and follicle-stimulating hormone (FSH), followed by downregulation of these hormones. This makes it effective in treating conditions such as prostate cancer, endometriosis, and central precocious puberty. It is typically administered via injection and is available in various formulations, including immediate-release and sustained-release forms.

Remarks

• The product complies with the specifications as per [Insert Pharmacopeia Standard, e.g., USP, EP, or JP].

• Storage conditions: Store at 2-8°C, protected from light and moisture.