CTX-012414 is a KAT6A inhibitor with IC50 value of 0.49 μM and KD value of 0.38 -M.
Uses
CTX-0124143 is a KAT6A inhibitor with a sulfonyl hydrazine skeleton[1].
References
[1] Duan Y, et al. Discovery of N-(2-oxoethyl) sulfanilamide-derived inhibitors of KAT6A (MOZ) against leukemia by an isostere strategy. Eur J Med Chem. 2023 Nov 15;260:115770. DOI:10.1016/j.ejmech.2023.115770
