育亨宾碱
育亨宾碱 用途与合成方法
Target | Value |
α2 adrenergic receptor
() | 12 nM(Ki) |
[ 3 H]Rauwolscine binding to α2 adrenergic receptor is reversible, stcreospccific, and saturable. [ 3 H]Rauwolscine specifically labels both the high and low affinity states of the α2 adrenergic receptor in brain membranes. [ 3 H]Rauwolscine also behaves as a 5-HT1A receptor agonist and this conclusion is compatible with earlier functional studies, indicating that rauwolscine (as well as yohimbine) has agonistic properties at the level of 5-HT autoreceptors. When using [ 3 H]5-HT as a radioligand, rauwolscine is determined to have relatively high affinity for the human receptor (K i human=14.3 nM, K i rat=35.8 nM). Saturation studies shows that the affinity of [ 3 H]Rauwolscine is similar in mouse, rat, rabbit, dog (2.33-3.03 nM) except man where it is significantly higher (0.98 nM) .
安全信息
危险品标志 | T |
---|---|
危险类别码 | 23/24/25 |
安全说明 | 22-36/37/39-45 |
危险品运输编号 | UN 1544 6.1/PG 2 |
WGK Germany | 3 |
RTECS号 | ZG1035000 |
危险等级 | 6.1 |
海关编码 | 29339900 |
育亨宾碱 价格(试剂级)
更新日期 | 产品编号 | 产品名称 | CAS号 | 包装 | 价格 |
---|---|---|---|---|---|
2024-11-08 | HY-12710 | 育亨宾碱 | 1 mg | 2320 | |
2024-11-08 | HY-12710 | 育亨宾碱 | 5 mg | 5800 |