(±)-
epi CP 47,497 is an analytical reference standard that is structurally categorized as a cannabinoid (CB). It is an epimer of (±)-CP 47,497 . (±)-CP 47,497 is a synthetic cannabinoid that avidly binds the CB
1 receptor (K
i = 2.2 nM) and is equivalent in analgesic potency to Δ
9-THC.
1,2 (±)-
epi CP 47,497 is regulated as a Schedule 1 drug in the United States. This product is intended for research and forensic applications.
[1] Huffman, J.W., Thompson, A.L.S., Wiley, J.L., et al. Synthesis and pharmacology of 1-deoxy analogs of CP-47,497 and CP-55,940 Bioorg. Med. Chem. 16(1),322-335(2008).
[2] Melvin, L.S., Milne, G.M., Johnson, M.R., et al. Structure-activity relationships for cannabinoid receptor-binding and analgesic activity: Studies of bicyclic cannabinoid analogs Mol. Pharmacol. 44(5),1008-1015(1993).