N-(Dicyclopropylmethyl)-4,5-dihydrooxazol-2-amin

Rilmenidine Chemische Eigenschaften,Einsatz,Produktion Methoden

• S-Sätze Betriebsanweisung:

  S22:Staub nicht einatmen.
  S24/25:Berührung mit den Augen und der Haut vermeiden.

• Beschreibung

  Rilmenidine is a new antihypertensive agent with a selective alphaz-agonist/antagonist profile, reportedly useful in the management of mild to moderate hypertension. Its fmt-line indication is possible because of the clear dissociation of its antihypertensive activity from other neurophannacological effects.

• Chemische Eigenschaften

  water soluble

• Originator

  Servier (France)

• Verwenden

  I1-imidazoline binding site ligand and a2-adrenoceptor agonist, exhibits higher I1 vs. a2 selectivity than clonidine

• Definition

  ChEBI: Rilmenidine is an isourea.

• Trademarks

  Hyperium

• Biologische Aktivität

  I 1 -imidazoline binding site selective ligand and α 2 -adrenoceptor agonist. Possesses greater I 1 vs α 2 selectivity than the prototypical compound, clonidine.

• Stoffwechselwegen

  In short-term rat hepatocyte cultures, oxaminozoline is metabolized and its four metabolites resulting from oxidation or hydrolysis are identified, three of which are identical to those reported in vivo. The presence of an additional minor metabolite in culture may be due to the higher metabolic rate of oxaminozoline in this model system.

Rilmenidine Upstream-Materialien And Downstream Produkte

N-(Dicyclopropylmethyl)-4,5-dihydrooxazol-2-amin Anbieter Lieferant Produzent Hersteller Vertrieb Händler.

Global(131)Suppliers

54187-04-1, Rilmenidine Verwandte Suche: