RLH 033 is a potent and selective ligand for the sigma 1 recognition site.
Uses
RLH-033 is a potent and selective ligand for the sigma 1 recognition site. RLH-033 has high affinity for sigma 1 sites labeled by [3H](+)-pentazocine with a Ki of 50 pM[1].
References
[1] R L Hudkins, et al. RLH-033, a novel, potent and selective ligand for the sigma 1 recognition site. Eur J Pharmacol. 1994 Dec 12;271(1):235-6. DOI:10.1016/0014-2999(94)90286-0
