5′-Guanidinonaltrindole di(trifluoroacetate) salt hydrate
TRC
G821700
1mg
$275
5′-Guanidinonaltrindole di(trifluoroacetate) salt hydrate
Properties
storage temp.
2-8°C
solubility
H2O: soluble30mg/mL
form
solid
Water Solubility
H2O: 30mg/mL
Description
5'-Guanidinonaltrindole di(trifluoroacetate)is a selective opioid receptor antagonist. GNTI is five-fold more potent and 500-fold more selective than norbinaltorphimine (nor-BNI) for the opioid receptor in smooth muscle preparations.