ChEBI: A benzodioxine that is idazoxan substituted at position 2 by a methoxy group.
Biological Activity
Potent, selective α 2 -adrenoceptor antagonist with very low affinity for imidazoline sites. Displays selectivity for the α 2D over the α 2A subtypes (pK d values are 9.7 and 8.2 respectively).
