SDZ SER 082 FUMARATE

SDZ SER 082 is a 5-HT2C and 5-HT2B receptor antagonist.

SDZ SER 082 Fumarate is a serotonin 2C receptor antagonist.

Selective 5-HT 2B/2C receptor antagonist with low affinity for 5-HT 1A receptors. Inhibits [ 3 H]-mesulergine binding to 5-HT 2C receptors with a pK D of 7.8. Inhibits 5-HT 2B mediated responses in the rat fundus (pK B = 7.34).