Anti-adrenergic (β-receptor).
Cicloprolol is a cardioselective beta-1 agonist. Itexhibitspartial agonist activity at the beta 1-adrenoceptor and beta 2-adrenoceptor. It has been suggested thatshort-term administration ofCicloprololis safe in moderate heart failure.
ChEBI: Cicloprolol is an aromatic ether.