SCH 50911 is a GABAB receptor antagonist.
A selective, competitive and orally active GABA B antagonist. Displays an IC 50 of 1.1 μ M at GABA B , approximately 60 times that of CGP 35348 ((3-Aminopropyl)(diethoxymethyl)phosphinic acid ) and no binding affinity for GABA A at concentrations up to 100 μ M.
SCH-50911 is a selective, competitive, orally active GABAB receptor antagonist.