アゴニスト阻害剤
- Structure:

- Chemical Name:フェンジリン塩酸塩
- CAS:13636-18-5
- MF:C23H26ClN
- Structure:

- Chemical Name:Acetic acid, 2-[4-[[4-(2-chlorophenyl)-2-thiazolyl]methoxy]-2-methylphenoxy]-
- CAS:1050506-75-6
- MF:C19H16ClNO4S
- Structure:

- Chemical Name:MK-0812
- CAS:624733-88-6
- MF:C24H34F3N3O3
- Structure:

- Chemical Name:VO-OHPIC 三水和物
- CAS:476310-60-8
- MF:C12H8N2O7V.3H2O
- Structure:

- Chemical Name:5-ブロモ-4'-クロロサリチルアニリド
- CAS:3679-64-9
- MF:C13H9BrClNO2
- Structure:

- Chemical Name:(2S,3R)-N-Hydroxy-N'-[(2S)-1-methylamino-1-oxo-3-phenylpropan-2-yl]-3-(2-methylpropyl)-2-(thiophen-2-ylsulfanylmethyl)butanediamide sodium salt
- CAS:130464-84-5
- MF:C23H32N3NaO4S2
- Structure:

- Chemical Name:セビパブリン
- CAS:849550-05-6
- MF:C18H18ClF5N6O
- Structure:

- Chemical Name:LY-335979
- CAS:167354-41-8
- MF:C32H31F2N3O2
- Structure:

- Chemical Name:CGS-21680 塩酸塩 水和物
- CAS:124182-57-6
- MF:C23H30ClN7O6
- Structure:

- Chemical Name:1-(2,6-ジフルオロベンジル)-3-フェニル-5-[フェニル(メチル)アミノメチル]-6-[p-(N′-メトキシウレイド)フェニル]チエノ[2,3-d]ピリミジン-2,4(1H,3H)-ジオン
- CAS:308831-61-0
- MF:C36H31F2N5O4S
- Structure:

- Chemical Name:[4-[(Hydroxyamino)carbonyl]phenyl]carbamic acid [6-[(diethylamino)methyl]-2-naphthalenyl]methyl ester
- CAS:497833-27-9
- MF:C24H27N3O4
- Structure:

- Chemical Name:ネロタンセリン
- CAS:839713-36-9
- MF:C18H15BrF2N4O2
- Structure:

- Chemical Name:4-メチル-3-((3-(2-(メチルアミノ)ピリミジン-4-イル)ピリジン-2-イル)オキシ)-N-(3-(トリフルオロメチル)フェニル)ベンズアミド
- CAS:870223-96-4
- MF:C25H20F3N5O2
- Structure:

- Chemical Name:LY-2608204
- CAS:1234703-40-2
- MF:C28H37N3O3S3
- Structure:

- Chemical Name:2-フルオロ-3-オキソ-4-メチル-N-[1H-イミダゾ[4,5-b]ピリジン-2-イルメチル]-4-アザ-5α-アンドロスタ-1-エン-17β-カルボアミド
- CAS:606101-58-0
- MF:C27H34FN5O2
- Structure:

- Chemical Name:テトラペプチド-61
- CAS:307297-39-8
- MF:C14H22N4O9
- Structure:

- Chemical Name:3-[[2-メトキシ-4-(フェニルアミノ)フェニル]アミノスルホニル]-2-チオフェンカルボン酸メチル
- CAS:1014691-61-2
- MF:C19H18N2O5S2
- Structure:

- Chemical Name:(3-Chlorophenyl)[3,4-dihydro-6,7-dimethoxy-1-[(4-methoxyphenoxy)methyl]-2(1H)-isoquinolinyl]methanone
- CAS:486427-17-2
- MF:C26H26ClNO5
- Structure:

- Chemical Name:N-(4-Acetyl-4,5-dihydro-5-methyl-5-phenyl-1,3,4-thiadiazol-2-yl)acetamide
- CAS:72926-24-0
- MF:C13H15N3O2S
- Structure:

- Chemical Name:N-(tert-Butyl)-3-[[5-methyl-2-[[4-(4-morpholinylmethyl)phenyl]amino]-4-pyrimidinyl]amino]benzenesulfonamide
- CAS:936091-15-5
- MF:C26H34N6O3S
- Structure:

- Chemical Name:3-(5-フルオロ-1H-インドール-3-イル)ピロリジン-2,5-ジオン
- CAS:198474-05-4
- MF:C12H9FN2O2
- Structure:

- Chemical Name:RK-20449
- CAS:364042-47-7
- MF:C29H34N6O
- Structure:

- Chemical Name:AZM475271
- CAS:476159-98-5
- MF:C23H27ClN4O3
- Structure:

- Chemical Name:ホスタマチニブ二ナトリウム六水和物
- CAS:914295-16-2
- MF:C23H24FN6Na2O9P
- Structure:

- Chemical Name:ビトペルチン
- CAS:845614-11-1
- MF:C21H20F7N3O4S
- Structure:

- Chemical Name:1-(2-メチルプロピル)-3-メチル-5-[[(4S)-4-ヒドロキシテトラヒドロイソオキサゾール-2-イル]カルボニル]-6-(3,5-ジメチル-1H-ピラゾール-4-イルメチル)チエノ[2,3-d]ピリミジン-2,4(1H,3H)-ジオン
- CAS:496791-37-8
- MF:C21H27N5O5S
- Structure:

- Chemical Name:PF-429242
- CAS:947303-87-9
- MF:C25H35N3O2
- Structure:

- Chemical Name:デラフロキサシン
- CAS:189279-58-1
- MF:C18H12ClF3N4O4
- Chemical Name:BMS-790052
- CAS:1214735-16-6
- MF:C40H50N8O6
- Structure:

- Chemical Name:シナシグアト
- CAS:329773-35-5
- MF:C36H39NO5
- Structure:

- Chemical Name:(S)-2-(2,6-ジクロロベンズアミド)-3-(2',6'-ジメトキシ-[1,1'-ビフェニル]-4-イル)プロパン酸
- CAS:232271-19-1
- MF:C24H21Cl2NO5
- Structure:

- Chemical Name:(3R,4S)-4-[[2-(5-フルオロ-2-ヒドロキシフェニル)-6,7-ジメトキシキナゾリン-4-イル]アミノ]-α,α-ジメチルピロリジン-3-メタノール
- CAS:1262849-73-9
- MF:C23H27FN4O4
- Structure:

- Chemical Name:SEA-0400
- CAS:223104-29-8
- MF:C21H19F2NO3
- Structure:

- Chemical Name:セジラニブマレイン酸塩
- CAS:857036-77-2
- MF:C25H27FN4O3·C4H4O4
- Structure:

- Chemical Name:ISX 9
- CAS:832115-62-5
- MF:C11H10N2O2S
- Structure:

- Chemical Name:オルテロネール
- CAS:566939-85-3
- MF:C18H17N3O2
- Structure:

- Chemical Name:ファトスタチン
- CAS:298197-04-3
- MF:C18H19BrN2S
- Structure:

- Chemical Name:R1487
- CAS:449808-64-4
- MF:C19H19ClF2N4O3
- Structure:

- Chemical Name:4-(4-(4-フルオロフェニル)-1-(ピペリジン-4-イル)-1H-イミダゾール-5-イル)-2-メトキシピリミジン
- CAS:193746-75-7
- MF:C19H20FN5O
- Structure:

- Chemical Name:2,5-Cyclohexadiene-1,4-dione, 2-Methyl-5-(1-Methylethyl)-, 1-oxiMe
- CAS:17302-61-3
- MF:C10H13NO2
- Structure:

- Chemical Name:ROCK-II inhibitor
- CAS:1273579-40-0
- MF:C24H28N4O4
- Structure:

- Chemical Name:N1-(4-クロロフェニル)-6-メチル-N5-[3-(9H-プリン-6-イル)-2-ピリジル]イソキノリン-1,5-ジアミン二塩酸塩
- CAS:1191385-19-9
- MF:C26H21Cl3N8
- Structure:

- Chemical Name:N-[(αS)-α-(ヒドロキシメチル)-3-クロロベンジル]-4-[2-[(2-クロロ-4-フルオロフェニル)アミノ]-5-メチル-4-ピリミジニル]-1H-ピロール-2-カルボアミド
- CAS:896720-20-0
- MF:C24H20Cl2FN5O2
- Structure:

- Chemical Name:BI605906
- CAS:960293-88-3
- MF:C17H22F2N4O3S2
- Structure:

- Chemical Name:BMS-687453
- CAS:1000998-59-3
- MF:C22H21ClN2O6
- Structure:

- Chemical Name:ELR-510444
- CAS:1233948-35-0
- MF:C19H16N2O2S2
- Structure:

- Chemical Name:Genz644282
- CAS:529488-28-6
- MF:C22H21N3O5
- Structure:

- Chemical Name:1-[1-(2-アミノ-4-ピリジニルメチル)-1H-インドール-4-イル]-3-(5-ブロモ-2-メトキシフェニル)尿素
- CAS:900573-88-8
- MF:C22H20BrN5O2
- Structure:

- Chemical Name:NS 11394
- CAS:951650-22-9
- MF:C23H19N3O
- Structure:

- Chemical Name:NVP-LCQ195
- CAS:902156-99-4
- MF:C17H19Cl2N5O4S
- Structure:

- Chemical Name:2-クロロ-4-[[(1R,2S)-1-[5-(4-シアノフェニル)-1,3,4-オキサジアゾール-2-イル]-2-ヒドロキシプロピル]アミノ]-3-メチルベンゾニトリル
- CAS:1182367-47-0
- MF:C20H16ClN5O2
- Structure:

- Chemical Name:SR 3335
- CAS:293753-05-6
- MF:C13H9F6NO3S2
- Structure:

- Chemical Name:テムサビル
- CAS:701213-36-7
- MF:C24H23N7O4
- Structure:

- Chemical Name:PF-543 (Citrate)
- CAS:1415562-83-2
- MF:C33H39NO11S
- Structure:

- Chemical Name:テトラエチル2,2',2'',2'''-(((3',6'-ジヒドロキシ-3-オキソ-3H-スピロ[イソベンゾフラン-1,9'-キサンテン]-4',5'-ジイル)ビス(メチレン))ビス(アザントリイル))テトラアセタート
- CAS:1170856-93-5
- MF:C38H42N2O13
- Structure:

- Chemical Name:B-Raf inhibitor 1
- CAS:1093100-40-3
- MF:C26H19ClN8
- Structure:

- Chemical Name:6-フルオロ-N-(4-フルオロベンジル)キナゾリン-4-アミン
- CAS:1262888-28-7
- MF:C15H11F2N3
- Structure:

- Chemical Name:(3E)-5-クロロ-3-({5-[3-(4-メチル-1,4-ジアゼパン-1-カルボニル)フェニル]フラン-2-イル}メチリデン)-1H-インドール-2-オン
- CAS:1202916-90-2
- MF:C26H24ClN3O3
- Structure:

- Chemical Name:FTI-277 トリフルオロアセタート塩
- CAS:170006-73-2
- MF:C22H29N3O3S2
- Structure:

- Chemical Name:STF31
- CAS:724741-75-7
- MF:C23H25N3O3S
- Structure:

- Chemical Name:GSK2838232
- CAS:1443461-21-9
- MF:C48H73ClN2O6
- Structure:

- Chemical Name:スペブルチニブベシル酸塩
- CAS:1360053-81-1
- MF:C28H28FN5O6S
- Structure:

- Chemical Name:タンジセルチブ
- CAS:899805-25-5
- MF:C21H23F3N6O2
- Structure:

- Chemical Name:KN93 hydrochloride
- CAS:1956426-56-4
- MF:C26H30Cl2N2O4S
- Structure:

- Chemical Name:イダロピルジン塩酸塩
- CAS:467458-02-2
- MF:C20H20ClF5N2O
- Structure:

- Chemical Name:1-[6-(3,5-ジクロロ-4-ヒドロキシフェニル)-4-[[4-[(ジメチルアミノ)メチル]シクロヘキシル]アミノ]-1,5-ナフチリジン-3-イル]エタノン
- CAS:1431697-89-0
- MF:C25H28Cl2N4O2
- Structure:

- Chemical Name:D 06
- CAS:256925-03-8
- MF:C23H24ClN3O2
- Structure:

- Chemical Name:Flumatinib mesylate
- CAS:895519-91-2
- MF:C30H33F3N8O4S
- Structure:

- Chemical Name:PF 02341066 hydrochloride
- CAS:1415560-69-8
- MF:C21H23Cl3FN5O
- Structure:

- Chemical Name:N-[2-Methyl-2-(2-phenyloxazol-4-yl)propyl]-3-[5-(trifluoroMethyl)-1,2,4-oxadiazol-3-yl]benzaMide
- CAS:1314891-22-9
- MF:C23H19F3N4O3
- Structure:

- Chemical Name:CNX-1351
- CAS:1276105-89-5
- MF:C30H35N7O3S
- Structure:

- Chemical Name:BenzenesulfonaMide, 3-chloro-2-Methyl-N-[5,6,7,8-tetrahydro-2-[(2-phenylethyl)aMino]-6-(phenylMethyl)pyrido[4,3-d]pyriMidin-4-yl]-
- CAS:1208123-85-6
- MF:C29H30ClN5O2S
- Structure:

- Chemical Name:2-(4,4-ジフルオロ-1-ピペリジニル)-N-(1-イソプロピル-4-ピペリジニル)-6-メトキシ-7-[3-(1-ピロリジニル)プロポキシ]キナゾリン-4-アミン
- CAS:1481677-78-4
- MF:C29H44F2N6O2
- Structure:

- Chemical Name:PCI 29732
- CAS:330786-25-9
- MF:C22H21N5O
- Structure:

- Chemical Name:LY900009
- CAS:209984-68-9
- MF:C23H27N3O4
- Structure:

- Chemical Name:SF1670(PTENinhibitor)
- CAS:345630-40-2
- MF:C19H17NO3
- Structure:

- Chemical Name:LEE011 (succinate hydrate)
- CAS:1374639-79-8
- MF:C27H36N8O5
- Structure:

- Chemical Name:アプロシテンタン
- CAS:1103522-45-7
- MF:C16H14Br2N6O4S
- Structure:

- Chemical Name:MI-773
- CAS:1303607-07-9
- MF:C29H34Cl2FN3O3
- Structure:

- Chemical Name:PLpro inhibitor
- CAS:1093070-14-4
- MF:C22H22N2O2
- Structure:

- Chemical Name:PNU-159682
- CAS:202350-68-3
- MF:C32H35NO13
- Structure:

- Chemical Name:FLLL32
- CAS:1226895-15-3
- MF:C28H32O6
- Structure:

- Chemical Name:GNF179
- CAS:1261114-01-5
- MF:C22H23ClFN5O
- Structure:

- Chemical Name:オマベロキソロン
- CAS:1474034-05-3
- MF:C33H44F2N2O3
- Structure:

- Chemical Name:Monohydroxy Netupitant
- CAS:910808-12-7
- MF:C30H32F6N4O2
- Structure:

- Chemical Name:LP 533401
- CAS:945976-43-2
- MF:C27H22F4N4O3
- Structure:

- Chemical Name:CID16020046
- CAS:834903-43-4
- MF:C25H19N3O4
- Structure:

- Chemical Name:HG6-64-1
- CAS:1315329-43-1
- MF:C32H34F3N5O2
- Structure:

- Chemical Name:KRCA-0008
- CAS:1472795-20-2
- MF:C30H37ClN8O4
- Structure:

- Chemical Name:リネリキシバット
- CAS:1345982-69-5
- MF:C28H38N2O7S
- Structure:

- Chemical Name:オリセリジン
- CAS:1401028-24-7
- MF:C22H30N2O2S
- Structure:

- Chemical Name:ベクラブビル
- CAS:958002-33-0
- MF:C36H45N5O5S
- Structure:

- Chemical Name:エルクサドリン
- CAS:864821-90-9
- MF:C32H35N5O5
- Structure:

- Chemical Name:LB-100
- CAS:1026680-07-8
- MF:C13H20N2O4
- Structure:

- Chemical Name:ソルシチニブ
- CAS:1206163-45-2
- MF:C22H23N5O2
- Structure:

- Chemical Name:2-(2-(3-クロロフェニル)ヒドラゾノ)-3-オキソ-3-(5-tert-ブチルイソオキサゾール-3-イル)プロパンニトリル
- CAS:263707-16-0
- MF:C16H15ClN4O2
- Structure:

- Chemical Name:TZ-9
- CAS:1002789-86-7
- MF:C17H14N6O4
- Structure:

- Chemical Name:3-Methyl-2-((1S,2S)-2-(quinolin-2-yl)cyclopropyl)-3H-iMidazo[4,5-f]quinoline
- CAS:1516896-09-5
- MF:C21H19N7
- Structure:

- Chemical Name:2-(2β-アミノシクロヘキサン-1β-イル)-4-(3-メチルフェニルアミノ)ピリミジン-5-カルボアミド
- CAS:1194961-19-7
- MF:C18H24N6O
