アゴニスト阻害剤
- Structure:

- Chemical Name:7-Chloro-9-oxo-9H-indeno[1,2-b]pyrazine-2,3-dicarbonitrile
- CAS:924296-39-9
- MF:C13H3ClN4O
- Structure:

- Chemical Name:(E)-(4R,9AS)-7-[3-メトキシ-4-(4-メチル-1H-イミダゾール-1-イル)ベンジリデン]-4-(3,4,5-トリフルオロフェニル)ヘキサヒドロピリド[2,1-C][1,4]オキサジン-6-オン
- CAS:937812-80-1
- MF:C26H24F3N3O3
- Structure:

- Chemical Name:N-[(3R)-2-オキソスピロ[1H-ピロロ[2,3-b]ピリジン-3(2H),2′(3′H)-[1H]インデン]-5′-イル]-2-[(8R)-6-オキソ-8-(3,5-ジフルオロフェニル)-7,10-ジアザスピロ[4.5]デカン-7-イル]アセトアミド
- CAS:957118-49-9
- MF:C31H29F2N5O3
- Structure:

- Chemical Name:MF-63
- CAS:892549-43-8
- MF:C23H11ClN4
- Structure:

- Chemical Name:N-[3-フルオロ-4-[(2-アミノ-3-クロロ-4-ピリジニル)オキシ]フェニル]-1-(4-フルオロフェニル)-2-オキソ-4-エトキシ-1,2-ジヒドロピリジン-3-カルボアミド
- CAS:1196681-44-3
- MF:C25H19ClF2N4O4
- Structure:

- Chemical Name:4-(1-ベンゾチオフェン-2-イル)-N-{4-[4-(ピロリジン-1-イル)ピペリジン-1-カルボニル]フェニル}ピリミジン-2-アミン
- CAS:1186195-62-9
- MF:C28H31ClN6OS
- Structure:

- Chemical Name:MCOPPB 三塩酸塩 水和物
- CAS:1028969-49-4
- MF:C26H40N4
- Structure:

- Chemical Name:VER-155008
- CAS:1134156-31-2
- MF:C25H23Cl2N7O4
- Structure:

- Chemical Name:CID 755673
- CAS:521937-07-5
- MF:C12H11NO3
- Structure:

- Chemical Name:4-アミノ-1-((2R,3R,4R,5R)-3-フルオロ-4-ヒドロキシ-5-(ヒドロキシメチル)-3-メチルテトラヒドロフラン-2-イル)ピリミジン-2(1H)-オン
- CAS:817204-33-4
- MF:C10H14FN3O4
- Structure:

- Chemical Name:クァルフロキシン
- CAS:865311-47-3
- MF:C35H33FN6O3
- Structure:

- Chemical Name:2-(5-(5-(4-(2-ブロモ-5-フルオロフェノキシ)ピペリジン-1-イル)-1,3,4-チアジアゾール-2-イル)-2H-テトラゾール-2-イル)酢酸
- CAS:1030612-87-3
- MF:C16H15BrFN7O3S
- Structure:

- Chemical Name:1-[4-(ジフェニルメチル)-1-ピペラジニル]-3,3-ジフェニル-1-プロパノン
- CAS:41332-24-5
- MF:C32H32N2O
- Structure:

- Chemical Name:N-[3-[[5-Cyclopropyl-2-[[3-(4-morpholinylmethyl)phenyl]amino]-4-pyrimidinyl]amino]propyl]cyclobutanecarboxamide
- CAS:1190378-57-4
- MF:C26H36N6O2
- Structure:

- Chemical Name:INCB 3284 diMesylate
- CAS:887401-93-6
- MF:C26H31F3N4O4
- Structure:

- Chemical Name:7-[3-(ジメチルアミノ)プロポキシ]-6-メトキシ-2-(4-メチル-1,4-ジアゼパン-1-イル)-N-(1-メチルピペリジン-4-イル)キナゾリン-4-アミン
- CAS:1197196-48-7
- MF:C26H43N7O2
- Structure:

- Chemical Name:シルベストロール
- CAS:697235-38-4
- MF:C34H38O13
- Structure:

- Chemical Name:TG100801
- CAS:867331-82-6
- MF:C33H30ClN5O3
- Structure:

- Chemical Name:2-シクロヘキシル-4-[(1-イソプロピルピペリジン-4-イル)アミノ]-6-メトキシ-7-[3-(ピロリジン-1-イル)プロポキシ]キナゾリン
- CAS:1255580-76-7
- MF:C30H47N5O2
- Structure:

- Chemical Name:テゴブビル
- CAS:1000787-75-6
- MF:C25H14F7N5
- Structure:

- Chemical Name:ポネシモド
- CAS:854107-55-4
- MF:C23H25ClN2O4S
- Structure:

- Chemical Name:3-PYRIDINECARBOXAMIDE, 6-(3-FLUOROPHENYL)-N-[1-(2,2,2-TRIFLUOROETHYL)-4-PIPERIDINYL]-
- CAS:1033836-12-2
- MF:C19H19F4N3O
- Structure:

- Chemical Name:N-(1H-ピロロ[2,3-c]ピリジン-5-イル)ベンズアミド
- CAS:300586-90-7
- MF:C14H11N3O
- Structure:

- Chemical Name:(alphaS)-3,5-difluoro-alpha-hydroxybenzeneacetic acid 2-(2-ethyl-4-hydroxy-3-methylbenzoyl)hydrazide
- CAS:1184940-46-2
- MF:C18H18F2N2O4
- Structure:

- Chemical Name:GNE-493
- CAS:1033735-94-2
- MF:C17H20N6O2S
- Structure:

- Chemical Name:フルエンスルホン
- CAS:318290-98-1
- MF:C7H5ClF3NO2S2
- Structure:

- Chemical Name:(Z)-2-decanoic acid
- CAS:15790-91-7
- MF:C10H18O2
- Structure:

- Chemical Name:N-(4-ブロモフェニル)-N′-(2,2,6,6-テトラメチル-4-ピペリジニル)オキサミド
- CAS:333352-59-3
- MF:C17H24BrN3O2
- Structure:

- Chemical Name:2-(2-クロロ-4-フルオロベンジル)-3-(4-フルオロフェニル)-7-(トリフルオロメチル)-2H-インダゾール
- CAS:875787-07-8
- MF:C21H12ClF5N2
- Structure:

- Chemical Name:5-{[2-メトキシ-4-(4-メチルピペラジン-1-イル)フェニル]アミノ}-2,9-ジメチル-2,4,6,9-テトラアザトリシクロ[9.4.0.03,8]ペンタデカ-1(15),3,5,7,11,13-ヘキサエン-10-オン
- CAS:1234479-76-5
- MF:C25H29N7O2
- Structure:

- Chemical Name:N-プロピル-4-(2-メチル-5-(シクロプロピルカルバモイル)アニリノ)-5-メチルピロロ[2,1-f][1,2,4]トリアジン-6-カルボアミド
- CAS:623152-17-0
- MF:C22H26N6O2
- Structure:

- Chemical Name:N-(3-ピリジニルメチル)-4-[プロパルギル[(2-メチル-4-オキソ-7-ブロモ-3,4-ジヒドロキナゾリン-6-イル)メチル]アミノ]ベンズアミド
- CAS:206275-15-2
- MF:C26H22BrN5O2
- Structure:

- Chemical Name:CM346 (OBENOXAZINE)
- CAS:173352-21-1
- MF:C15H21N3O2S
- Structure:

- Chemical Name:(3R)-3-(モルホリノカルボニル)-1′-(9-アントラセニルカルボニル)-1,4′-ビピペリジン
- CAS:591778-68-6
- MF:C30H35N3O3
- Structure:

- Chemical Name:(S)-2-[[[2β-ベンジル-3-オキソ-4-[(5-メチル-1H-イミダゾール-4-イル)メチル]ピペラジノ]カルボニル]アミノ]-4-メチルペンタン酸
- CAS:501010-06-6
- MF:C23H31N5O4
- Structure:

- Chemical Name:2-シクロヘキシル-N-(3,4-ジクロロフェニル)-1H-イミダゾ[4,5-c]キノリン-4-アミン
- CAS:890087-21-5
- MF:C22H20Cl2N4
- Structure:

- Chemical Name:MC 976
- CAS:129831-99-8
- MF:C27H42O3
- Structure:

- Chemical Name:NMS-P715
- CAS:1202055-34-2
- MF:C35H42N8O3
- Structure:

- Chemical Name:GC1
- CAS:211110-63-3
- MF:C20H24O4
- Structure:

- Chemical Name:1-(2-ブロモフェニル)-3-[(3S)-1-[5-(トリフルオロメチル)-2-ピリジル]-3-ピロリジニル]尿素
- CAS:501951-42-4
- MF:C17H16BrF3N4O
- Structure:

- Chemical Name:TH 237A
- CAS:935467-97-3
- MF:C18H17F2NO3
- Structure:

- Chemical Name:N-メシチル-4-メトキシベンゼンスルホンアミド
- CAS:349085-82-1
- MF:C16H19NO3S
- Structure:

- Chemical Name:CID-2858522
- CAS:758679-97-9
- MF:C28H39N3O3
- Structure:

- Chemical Name:JW55
- CAS:664993-53-7
- MF:C25H26N2O5
- Structure:

- Chemical Name:WAY-161503
- CAS:75704-24-4
- MF:C11H11Cl2N3O
- Structure:

- Chemical Name:BPTES
- CAS:314045-39-1
- MF:C24H24N6O2S3
- Structure:

- Chemical Name:2-[8-[2-(ベンゾチアゾール-2-イル)ヒドラゾノ]-5,6,7,8-テトラヒドロナフタレン-2-イル]-5-[3-[4-(アミノメチル)フェノキシ]プロピル]チアゾール-4-カルボン酸
- CAS:1431866-33-9
- MF:C31H29N5O3S2
- Structure:

- Chemical Name:3-[(1S,2S)-2-Hydroxycyclohexyl]-6-[(6-methyl-3-pyridinyl)methyl]benzo[h]quinazolin-4(3H)-one
- CAS:1227923-29-6
- MF:C25H25N3O2
- Structure:

- Chemical Name:GSK-525768A
- CAS:1260530-25-3
- MF:C22H22ClN5O2
- Structure:

- Chemical Name:JNK inhibitor
- CAS:1408064-71-0
- MF:C28H27N7O2
- Structure:

- Chemical Name:グラゾプレビル水和物
- CAS:1350462-55-3
- MF:C38H50N6O9S.H2O
- Structure:

- Chemical Name:MonoMethyl Dolastatin 10
- CAS:203849-91-6
- MF:C41H66N6O6S
- Structure:

- Chemical Name:SB408124 Hydrochloride
- CAS:1431697-90-3
- MF:C19H19ClF2N4O
- Structure:

- Chemical Name:{4-[(2S)-5-(カルバモイルアミノ)-2-[(2S)-2-[6-(2,5-ジオキソ-2,5-ジヒドロ-1H-ピロール-1-イル)ヘキサンアミド]-3-メチルブタンアミド]ペンタンアミド]フェニル}メチルN-[(1S)-1-{[(1S)-1-{[(3R,4S,5S)-1-[(2S)-2-[(1R,2R)-2-{[(1S,2R)-1-ヒドロキシ-1-フェニルプロパン-2-イル]カルバモイル}-1-メトキシ-2-メチルエチル]ピロリジン-1-イル]-3-メトキシ-5-メチル-1-オキソヘプタン-4-イル](メチル)カルバモイル}-2-メチルプロピル]カルバモイル}-2-メチルプロピル]-N-メチルカルバマート
- CAS:646502-53-6
- MF:C68H105N11O15
- Structure:

- Chemical Name:1,4-フェニレンビス(1,4'-ビピペリジン-1'-イルメタノン)
- CAS:1418741-86-2
- MF:C28H42N4O2
- Structure:

- Chemical Name:AZ 876
- CAS:898800-26-5
- MF:C24H29N3O3S
- Structure:

- Chemical Name:(23S)-6α-エチル-7α,12α-ジヒドロキシ-23-メチル-5β-コラン-24-酸
- CAS:1199796-29-6
- MF:C27H46O5
- Structure:

- Chemical Name:エリグルスタット酒石酸塩
- CAS:928659-70-5
- MF:C50H78N4O14
- Structure:

- Chemical Name:5-フルオロ-N-(3-ヒドロキシベンジル)-1H-インドール-2-カルボキサミド
- CAS:518058-84-9
- MF:C16H13FN2O2
- Structure:

- Chemical Name:SRPIN340
- CAS:218156-96-8
- MF:C18H18F3N3O
- Structure:

- Chemical Name:Lパ2アンタゴニスト1
- CAS:1017606-66-4
- MF:C20H23Cl2N5O2S2
- Structure:

- Chemical Name:GDC 0068 (Hydrochloride)
- CAS:1396257-94-5
- MF:C24H33Cl2N5O2
- Structure:

- Chemical Name:Finasteride (acetate)
- CAS:222989-99-3
- MF:C25H40N2O4
- Structure:

- Chemical Name:1-(3-メトキシベンジル)-3-(4-(ピリジン-4-イル)チアゾール-2-イル)尿素
- CAS:1342276-76-9
- MF:C17H16N4O2S
- Structure:

- Chemical Name:YLF-466D
- CAS:1273323-67-3
- MF:C29H20ClNO3
- Structure:

- Chemical Name:オマダサイクリントシル酸塩
- CAS:1075240-43-5
- MF:C36H48N4O10S
- Structure:

- Chemical Name:9-[2-フルオロ-3-(3-メトキシフェニルアミノ)プロピル]-3,6-ジブロモ-9H-カルバゾール
- CAS:1235481-90-9
- MF:C22H19Br2FN2O
- Structure:

- Chemical Name:STF083010
- CAS:307543-71-1
- MF:C15H11NO3S2
- Structure:

- Chemical Name:TUG891
- CAS:1374516-07-0
- MF:C23H21FO3
- Structure:

- Chemical Name:(3Z)-3-[α-[[4-[メチル[2-(4-メチルピペラジノ)アセチル]アミノ]フェニル]アミノ]ベンジリデン]-2-オキソ-1H-インドール-6-カルボン酸
- CAS:894783-71-2
- MF:C30H31N5O4
- Structure:

- Chemical Name:DUBs-IN-2
- CAS:924296-19-5
- MF:C15H9N5O
- Structure:

- Chemical Name:ソリスロマイシン
- CAS:760981-83-7
- MF:C43H65FN6O10
- Structure:

- Chemical Name:トスフロキサシントシル酸塩水和物
- CAS:1400591-39-0
- MF:C26H23F3N4O6S
- Structure:

- Chemical Name:AR7
- CAS:80306-38-3
- MF:C15H12ClNO
- Structure:

- Chemical Name:c-di-AMP
- CAS:54447-84-6
- MF:C20H24N10O12P2
- Structure:

- Chemical Name:CPI-169
- CAS:1450655-76-1
- MF:C27H36N4O5S
- Structure:

- Chemical Name:Helioxanthin 8-1
- CAS:840529-13-7
- MF:C20H12N2O6
- Structure:

- Chemical Name:HTH-01-015
- CAS:1613724-42-7
- MF:C26H28N8O
- Structure:

- Chemical Name:Mutated EGFR-IN-1
- CAS:1421372-66-8
- MF:C25H31N7O
- Structure:

- Chemical Name:1α-(4-クロロフェニル)-2-[4-[メチル[[4-(3-オキソ-4-メチルピペラジノ)シクロヘキシル]メチル]アミノ]フェニル]-6-メトキシ-7-イソプロポキシ-1,2-ジヒドロイソキノリン-3(4H)-オン
- CAS:1313363-54-0
- MF:C38H47ClN4O4
- Structure:

- Chemical Name:(1R,4R)-4-(2-(ブチルアミノ)-5-(4-((4-メチルピペラジン-1-イル)メチル)フェニル)-7H-ピロロ[2,3-D]ピリミジン-7-イル)シクロヘキサノール
- CAS:1429881-91-3
- MF:C28H40N6O
- Structure:

- Chemical Name:2-[(3S)-3β-(2-ピリジニルメトキシ)ピロリジノ]-5-(トリフルオロメチル)安息香酸
- CAS:1515856-92-4
- MF:C18H17F3N2O3
- Structure:

- Chemical Name:AZ191
- CAS:1594092-37-1
- MF:C24H27N7O
- Structure:

- Chemical Name:ピミテスピブ
- CAS:1260533-36-5
- MF:C25H26N8O
- Structure:

- Chemical Name:CID 797718
- CAS:370586-05-3
- MF:C12H11NO3
- Structure:

- Chemical Name:2-[(2S)-1-(tert-ブチルオキシカルボニル)-2-ピロリジニル]チアゾール-4-カルボン酸
- CAS:251349-54-9
- MF:C13H18N2O4S
- Structure:

- Chemical Name:ARRY-614
- CAS:945614-12-0
- MF:C31H33FN6O3
- Structure:

- Chemical Name:5-TERT-ブチルトキシキナゾリン-2,4-ジアミン
- CAS:1009734-33-1
- MF:C12H16N4O
- Structure:

- Chemical Name:N-ベンジル-N-メチル-1-(4-(トリフルオロメチル)ベンジル)ピペリジン-3-カルボキサミド
- CAS:1350920-22-7
- MF:C22H25F3N2O
- Structure:

- Chemical Name:N-(3-(5-(2-hydroxypropan-2-yl)-1,2,4-oxadiazol-3-yl)benzyl)-2-(pyridin-2-yl)pyriMidine-5-carboxaMide
- CAS:1234708-04-3
- MF:C22H20N6O3
- Structure:

- Chemical Name:7-[ベンジル(メチル)アミノ]-2-オキソ-2H-クロメン-3-カルボン酸
- CAS:1472624-85-3
- MF:C18H15NO4
- Structure:

- Chemical Name:レシヌラドナトリウム
- CAS:1151516-14-1
- MF:C17H13BrN3O2S.Na
- Structure:

- Chemical Name:LY-2584702 (hydrochloride)
- CAS:1082948-81-9
- MF:C21H20ClF4N7
- Structure:

- Chemical Name:ミベブレシブ
- CAS:1445993-26-9
- MF:C22H19F2N3O4S
- Structure:

- Chemical Name:CZC-54252
- CAS:1191911-27-9
- MF:C22H25ClN6O4S
- Structure:

- Chemical Name:8-(3,5-ジクロロフェニルチオ)-9-[3-(イソプロピルアミノ)プロピル]-9H-プリン-6-アミン
- CAS:1454619-14-7
- MF:C17H20Cl2N6S
- Structure:

- Chemical Name:2-(1-Phenyl-cyclopropylamino)-pyrimidine-5-carboxylic acid hydroxyamide
- CAS:1375465-91-0
- MF:C14H14N4O2
- Structure:

- Chemical Name:N-methyl-3-(1-(4-(piperazin-1-yl)phenyl)-5-(4'-(trifluoromethyl)-[1,1'-biphenyl]-4-yl)-1H-pyrazol-3-yl)propanamide
- CAS:1333146-24-9
- MF:C30H30F3N5O
- Structure:

- Chemical Name:4-メチル-1-(1H-ピラゾール-4-イルメチル)-5-[(4-{[6-(2,2,2-トリフルオロエチル)チエノ[2,3-d]ピリミジン-4-イル]アミノ}ピペリジン-1-イル)メチル]インドール-2-カルボニトリル
- CAS:1857417-13-0
- MF:C28H27F3N8S
- Structure:

- Chemical Name:パリタプレビル
- CAS:1216941-48-8
- MF:C40H43N7O7S