インヒビター
免疫抑制剤
タンパク質チロシンキナーゼ
神経シグナル伝達経路(神経シグナリング)
PI3K / AKT / mTOR阻害剤(PI3K / AKT / mTORの)
代謝(代謝)
細胞周期(細胞周期)
エピジェネティクス(エピジェネティクス)
細胞骨格(細胞骨格シグナリング)
血管新生(血管新生)
DNA損傷(DNA損傷)
プロテアソーム(プロテアーゼ)
アポトーシス(アポトーシス)
マイトジェン活性化プロテインキナーゼ(MAPK)
内分泌ホルモン(内分泌学&ホルモン)
Gタンパク質共役受容体(GPCRおよびGタンパク質)
膜貫通トランスポーター(膜貫通トランスポーター)
タンパク質チロシンキナーゼ/シグナル伝達物質および転写インヒビターの活性化因子(JAK / STAT)
TGF-β/ Smadのシグナル伝達経路阻害剤(TGF-β/ Smadの)
幹細胞とWntシグナル伝達経路(細胞&Wntシグナル幹)
核転写因子(NF-κB)
ユビキチン化阻害剤(ユビキチン)
微生物(微生物学)
オートファジーリソソーム(オートファジー)
- Structure:
- Chemical Name:FGFR inhibitor
- CAS:848318-25-2
- MF:C18H15N2NaO4
- Structure:
- Chemical Name:WAY-600
- CAS:1062159-35-6
- MF:C28H30N8O
- Structure:
- Chemical Name:C-646
- CAS:328968-36-1
- MF:C24H19N3O6
- Structure:
- Chemical Name:1-(アミノメチル)シクロヘキサン酢酸・塩酸塩
- CAS:60142-95-2
- MF:C9H12ClD6NO2
- Structure:
- Chemical Name:6-(2-Chloro-4-thiazol-5-yl-phenyl)-8-ethyl-2-[4-(4-Methyl-piperazin-1-yl)-phenylaMino]-8H-pyrido[2,3-d]pyriMidin-7-one
- CAS:1286739-19-2
- MF:C29H28ClN7OS
- Structure:
- Chemical Name:4-[4-(5-ニトロフラン-2-イルメチレン)-3,5-ジオキソピラゾリジン-1-イル]安息香酸エチル
- CAS:418805-02-4
- MF:C17H13N3O7
- Structure:
- Chemical Name:2-[[4-[1-(2,2,2-トリフルオロエチル)-4-(4-ピリジル)-1H-ピラゾール-3-イル]フェノキシ]メチル]キノリン
- CAS:1292799-56-4
- MF:C25H20N4O
- Structure:
- Chemical Name:(Z)-3-(3-(3,5-bis(trifluoroMethyl)phenyl)-1H-1,2,4-triazol-1-yl)-1-(3,3-
- CAS:1421919-75-6
- MF:C16H10F8N4O
- Structure:
- Chemical Name:2-[[(4-フェノキシフェニル)スルホニル]メチル]チイラン
- CAS:292605-14-2
- MF:C15H14O3S2
- Structure:
- Chemical Name:{3-[(4-クロロフェニル)スルファニル]-4-アセトアミド-2-メチルインドール-1-イル}酢酸
- CAS:802904-66-1
- MF:C19H17ClN2O3S
- Structure:
- Chemical Name:エントスプレチニブ
- CAS:1229208-44-9
- MF:C23H21N7O
- Structure:
- Chemical Name:CCG-1423
- CAS:285986-88-1
- MF:C18H13ClF6N2O3
- Structure:
- Chemical Name:ML133塩酸塩
- CAS:1222781-70-5
- MF:C19H20ClNO
- Structure:
- Chemical Name:LDN193189 塩酸塩
- CAS:1062368-62-0
- MF:C25H23ClN6
- Structure:
- Chemical Name:1,1′-ジチオビス(2-ナフトール)
- CAS:42521-82-4
- MF:C20H14O2S2
- Structure:
- Chemical Name:KU 0060648
- CAS:881375-00-4
- MF:C33H34N4O4S
- Structure:
- Chemical Name:N-[5-(ピラジン-2-イル)-2-ピリジニル]-2-(2′,3-ジメチル-2,4′-ビピリジン-5-イル)アセトアミド
- CAS:1243244-14-5
- MF:C23H20N6O
- Structure:
- Chemical Name:GSK2656157
- CAS:1337532-29-2
- MF:C23H21FN6O
- Structure:
- Chemical Name:エラスティン
- CAS:571203-78-6
- MF:C30H31ClN4O4
- Structure:
- Chemical Name:4-(6-メトキシ-2-ナフチル)-2-(4-メチルスルフィニルフェニル)-5-(4-ピリジル)-1H-イミダゾール
- CAS:948557-43-5
- MF:C26H21N3O2S
- Structure:
- Chemical Name:AZD 9668
- CAS:848141-11-7
- MF:C25H22F3N5O4S
- Structure:
- Chemical Name:ベルジネクソル
- CAS:1392136-43-4
- MF:C18H12F6N6O
- Structure:
- Chemical Name:4-(6-((4-(シクロプロピルメチル)ピペラジン-1-イル)メチル)-2-(5-フルオロ-1H-インドール-4-イル)チエノ[3,2-D]ピリミジン-4-イル)モルホリン
- CAS:955977-50-1
- MF:C27H31FN6OS
- Structure:
- Chemical Name:EHT1864
- CAS:754240-09-0
- MF:C25H27F3N2O4S2HCl
- Structure:
- Chemical Name:バルリチニブ
- CAS:845272-21-1
- MF:C22H19ClN6O2S
- Structure:
- Chemical Name:MELDONIUM 二水和物
- CAS:86426-17-7
- MF:C6H14N2O2.2H2O
- Structure:
- Chemical Name:N-[[(2R)-1,4-ジオキサン-2-イル]メチル]-N-メチル-N′-[3-(1-メチル-1H-ピラゾール-4-イル)-5-オキソ-5H-ベンゾ[4,5]シクロヘプタ[1,2-b]ピリジン-7-イル]スルファミド
- CAS:917879-39-1
- MF:C24H25N5O5S
- Structure:
- Chemical Name:LB 42708
- CAS:226929-39-1
- MF:C30H27BrN4O2
- Structure:
- Chemical Name:NSC23766
- CAS:1177865-17-6
- MF:C24H35N7
- Structure:
- Chemical Name:VER-50589
- CAS:747413-08-7
- MF:C19H17ClN2O5
- Structure:
- Chemical Name:N-[(1β,5β)-8-[5-(シクロプロピルカルボニル)-2-ピリジニル]-8-アザビシクロ[3.2.1]オクタン-3α-イル]-2-メチル-5-[[(R)-sec-ブチル]アミノ]-1,4-ベンゼンジカルボアミド
- CAS:1149705-71-4
- MF:C29H37N5O3
- Structure:
- Chemical Name:MI-2 (Menin-MLL Inhibitor)
- CAS:1271738-62-5
- MF:C18H25N5S2
- Structure:
- Chemical Name:CAY10603
- CAS:1045792-66-2
- MF:C22H30N4O6
- Structure:
- Chemical Name:HO-3867
- CAS:1172133-28-6
- MF:C28H30F2N2O2
- Structure:
- Chemical Name:2,6-ジブロモ-4-[(6,7-ジメトキシキナゾリン-4-イル)アミノ]フェノール
- CAS:211555-05-4
- MF:C16H13Br2N3O3
- Structure:
- Chemical Name:4,4'-(1-メチルエチレン)ビス(2,6-ピペラジンジオン)
- CAS:21416-67-1
- MF:C11H16N4O4
- Structure:
- Chemical Name:E-3810
- CAS:1058137-23-7
- MF:C26H25N3O4
- Structure:
- Chemical Name:BAM7
- CAS:331244-89-4
- MF:C21H19N5O2S
- Structure:
- Chemical Name:DCC-2618
- CAS:1225278-16-9
- MF:C26H21F2N5O3
- Structure:
- Chemical Name:pf-5274857
- CAS:1373615-35-0
- MF:C20H25ClN4O3S
- Structure:
- Chemical Name:3-[[2-(2-ピリジル)-6-(1,2,4,5-テトラヒドロ-3H-3-ベンゾアゼピン-3-イル)-4-ピリミジニル]アミノ]プロピオン酸エチル
- CAS:1373423-53-0
- MF:C24H27N5O2
- Structure:
- Chemical Name:ZM39923塩酸塩
- CAS:1021868-92-7
- MF:C23H26ClNO
- Structure:
- Chemical Name:NSC697923
- CAS:343351-67-7
- MF:C11H9NO5S
- Structure:
- Chemical Name:4-[(2S)-1-アセチル-2β-メチル-4β-[(4-クロロフェニル)アミノ]-1,2,3,4-テトラヒドロキノリン-6-イル]安息香酸
- CAS:1300031-52-0
- MF:C25H23ClN2O3
- Structure:
- Chemical Name:(3S)-1-(4-フルオロベンゾイル)-3-[3-(4-フルオロフェニル)-1,2,4-オキサジアゾール-5-イル]ピペリジン
- CAS:851881-60-2
- MF:C20H17F2N3O2
- Structure:
- Chemical Name:CAY10505
- CAS:1218777-13-9
- MF:C14H8FNO3S
- Structure:
- Chemical Name:N-(3-アミノプロピル)-N-[(S)-1-[7-クロロ-3-ベンジル-4-オキソ-3,4-ジヒドロキナゾリン-2-イル]-3-ブチニル]-3-クロロ-2-フルオロベンズアミド
- CAS:1095253-39-6
- MF:C28H24Cl2FN5O2
- Structure:
- Chemical Name:PIK-293
- CAS:900185-01-5
- MF:C22H19N7O
- Structure:
- Chemical Name:TG 100713
- CAS:925705-73-3
- MF:C12H10N6O
- Structure:
- Chemical Name:SBE 13 塩酸塩
- CAS:1052532-15-6
- MF:C24H28Cl2N2O4
- Structure:
- Chemical Name:デファクチニブ
- CAS:1073154-85-4
- MF:C20H21F3N8O3S
- Structure:
- Chemical Name:N-(6-{4-[({4-[(4-メチルピペラジン-1-イル)メチル]-3-(トリフルオロメチル)フェニル}カルバモイル)メチル]フェノキシ}ピリミジン-4-イル)シクロプロパンカルボキサミド
- CAS:1421227-53-3
- MF:C29H31F3N6O3
- Structure:
- Chemical Name:N-[3-[[5-クロロ-2-[[2-メトキシ-4-(4-メチル-1-ピペラジニル)フェニル]アミノ]-4-ピリミジニル]オキシ]フェニル]プロパンアミド
- CAS:1214265-58-3
- MF:C25H29ClN6O3
- Structure:
- Chemical Name:GSK-LSD1
- CAS:1431368-48-7
- MF:C14H20N2
- Structure:
- Chemical Name:AKT Kinase Inhibitor
- CAS:842148-40-7
- MF:C16H19N7O3
- Structure:
- Chemical Name:RGFP 109
- CAS:1215493-56-3
- MF:C20H25N3O2
- Structure:
- Chemical Name:カボテグラビル
- CAS:1051375-10-0
- MF:C19H17F2N3O5
- Structure:
- Chemical Name:2-(ベンゾイルアミノ)-1-(3-フェニルプロピル)-1H-ベンゾイミダゾール-5-カルボン酸メチル
- CAS:1374601-40-7
- MF:C25H23N3O3
- Structure:
- Chemical Name:LDC1267
- CAS:1361030-48-9
- MF:C30H26F2N4O5
- Structure:
- Chemical Name:N-エチル-3-(2,4-ジヒドロキシ-5-クロロフェニル)-4-(4-メトキシフェニル)-1H-ピラゾール-5-カルボアミド
- CAS:940289-57-6
- MF:C19H18ClN3O4
- Structure:
- Chemical Name:マレイン酸WAY-100635
- CAS:1092679-51-0
- MF:C29H38N4O6
- Structure:
- Chemical Name:LDC000067
- CAS:1073485-20-7
- MF:C18H18N4O3S
- Structure:
- Chemical Name:Raf265 derivative
- CAS:1942849-27-5
- MF:C23H14F6N6O
- Structure:
- Chemical Name:LMK235
- CAS:1418033-25-6
- MF:C15H22N2O4
- Structure:
- Chemical Name:Cathepsin Inhibitor 1
- CAS:225120-65-0
- MF:C20H24ClN5O2
- Structure:
- Chemical Name:Deltarasin
- CAS:1440898-61-2
- MF:C40H37N5O
- Structure:
- Chemical Name:アフレセルチブ
- CAS:1047644-62-1
- MF:C18H17Cl2FN4OS
- Structure:
- Chemical Name:BS-181 HCl
- CAS:1397219-81-6
- MF:C22H33ClN6
- Structure:
- Chemical Name:RGFP966
- CAS:1396841-57-8
- MF:C21H19FN4O
- Structure:
- Chemical Name:ReModelin hydrobroMide
- CAS:1622921-15-6
- MF:C15H15BrN4S
- Structure:
- Chemical Name:WIKI4
- CAS:838818-26-1
- MF:C29H23N5O3S
- Structure:
- Chemical Name:FTI-277 トリフルオロアセタート塩
- CAS:180977-34-8
- MF:C22H30ClN3O3S2
- Structure:
- Chemical Name:PD-151746
- CAS:179461-52-0
- MF:C11H8FNO2S
- Structure:
- Chemical Name:3-アミノ-4-(シクロヘキシルアミノ)安息香酸エチル
- CAS:347174-05-4
- MF:C15H22N2O2
- Structure:
- Chemical Name:IEM 1754 dihydrobroMide
- CAS:162831-31-4
- MF:C16H32Br2N2
- Structure:
- Chemical Name:2-[[2-(2-メトキシ-4-モルホリン-4-イルフェニル)アミノ-5-(トリフルオロメチル)ピリジン-4-イル]アミノ]-N-メチルベンズアミド
- CAS:1061353-68-1
- MF:C25H26F3N5O3
- Structure:
- Chemical Name:Tubastatin-A
- CAS:1252003-15-8
- MF:C20H21N3O2
- Structure:
- Chemical Name:AGK-2
- CAS:304896-28-4
- MF:C23H13Cl2N3O2
- Structure:
- Chemical Name:MI-3 (Menin-MLL Inhibitor)
- CAS:1271738-59-0
- MF:C18H25N5S2
- Structure:
- Chemical Name:2-[(9S)-7-(4-クロロフェニル)-4,5,13-トリメチル-3-チア-1,8,11,12-テトラアザトリシクロ[8.3.0.02,6]トリデカ-2(6),4,7,10,12-ペンタエン-9-イル]アセトアミド
- CAS:1446144-04-2
- MF:C19H18ClN5OS
- Structure:
- Chemical Name:4-((2-(((1R,2R)-2-ヒドロキシシクロヘキシル)アミノ)ベンゾ[D]チアゾール-6-イル)オキシ)-N-メチルピコリンアミド
- CAS:953769-46-5
- MF:C20H22N4O3S
- Structure:
- Chemical Name:AZD 2932
- CAS:883986-34-3
- MF:C24H25N5O4
- Structure:
- Chemical Name:LFM-A13
- CAS:244240-24-2
- MF:C11H8Br2N2O2
- Structure:
- Chemical Name:BMX-IN-1
- CAS:1431525-23-3
- MF:C29H24N4O4S
- Structure:
- Chemical Name:N,N′-(1,6-ヘキサンジイル)-Nα,Nα′-ビス[[(2S)-1-[(2S)-2-[(N-メチル-L-Ala-)アミノ]-2-シクロヘキシルアセチル]-2-ピロリジニル]カルボニル]ビス(L-フェニルアラニンアミド)
- CAS:1001600-56-1
- MF:C70H96N10O8
- Structure:
- Chemical Name:シポニモド
- CAS:1230487-00-9
- MF:C29H35F3N2O3
- Structure:
- Chemical Name:1-(2-ヒドロキシフェニル)3-[(1R,4R)-5-(2-ピリジニル)-2,5-ジアザビシクロ[2.2.1]ヘプタン-2-イル]-2-プロペン-1-オン
- CAS:1819363-80-8
- MF:C19H19N3O2
- Structure:
- Chemical Name:PFI-2
- CAS:1627676-59-8
- MF:C23H25F4N3O3S
- Structure:
- Chemical Name:MG149
- CAS:1243583-85-8
- MF:C22H28O3
- Structure:
- Chemical Name:4-[6-アミノ-4-(5-クロロ-1H,3H-ナフト[1,8-cd]ピラン-6-イル)-1,3,5-トリアジン-2-イルチオ]ブタンアミド
- CAS:959763-06-5
- MF:C19H18ClN5O2S
- Structure:
- Chemical Name:ISRIB (trans-isoMer)
- CAS:1597403-47-8
- MF:C22H24Cl2N2O4
- Structure:
- Chemical Name:サンタクルツマートA
- CAS:1477949-42-0
- MF:C15H22N2O3
- Structure:
- Chemical Name:BenzaMide, N-[4-[(4-ethyl-1-piperazinyl)Methyl]-3-(trifluoroMethyl)phenyl]-4-Methyl-3-[[[5-(2-thienyl)-3-pyridinyl]carbonyl]aMino]-
- CAS:1186206-79-0
- MF:C32H32F3N5O2S
- Structure:
- Chemical Name:GZD824
- CAS:1421783-64-3
- MF:C31H35F3N6O7S2
- Structure:
- Chemical Name:YH239-EE
- CAS:1364488-67-4
- MF:C25H27Cl2N3O4
- Structure:
- Chemical Name:Triapine
- CAS:200933-27-3
- MF:C7H9N5S
- Structure:
- Chemical Name:BIX 01294三塩酸塩水和物
- CAS:1392399-03-9
- MF:C28H41Cl3N6O2
- Structure:
- Chemical Name:K-Ras inhibitor
- CAS:1469338-01-9
- MF:C20H30ClN3O2S3
- Structure:
- Chemical Name:3-(3,4,5-トリメトキシフェニル)-2-メチル-5-(4-ピペラジノフェニル)ピリジン
- CAS:1627503-67-6
- MF:C25H29N3O3
- Structure:
- Chemical Name:SH-4-54
- CAS:1456632-40-8
- MF:C29H27F5N2O5S