Inhibitor Activator
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- Structure:

- Chemical Name:BTdCPU
- CAS:1257423-87-2
- MF:C13H8Cl2N4OS
- Structure:

- Chemical Name:Pyridazine, 3-[[(2-chloro-6-fluorophenyl)methyl]thio]-6-(2-pyridinyl)-
- CAS:892415-28-0
- MF:C16H11ClFN3S
- Chemical Name:[oxido-(2,3,4,5,6-pentaphosphonatooxycyclohexyl)oxyphosphoryl] phosphate
- CAS:193743-89-4
- MF:
- Structure:

- Chemical Name:EG-011
- CAS:2377113-41-0
- MF:C28H26N4O4
- Structure:

- Chemical Name:(1E,4E)-1,5-Bis(2-Methoxyphenyl)penta-1,4-dien-3-one
- CAS:39777-61-2
- MF:C19H18O3
- Chemical Name:WS3 (IΚB/IKK inhibitor)
- CAS:
- MF:
- Chemical Name:PND-1186 (FAK inhibitor)
- CAS:
- MF:
- Chemical Name:PI-103 (PI3K inhibitor)
- CAS:
- MF:
- Chemical Name:PFI-4 (EPIGENETIC READER DOMAIN inhibitor)
- CAS:
- MF:
- Chemical Name:PANOBINOSTAT (LBH589) (HDAC inhibitor)
- CAS:
- MF:
- Chemical Name:OSELTAMIVIR ACID (NEURAMINIDASE Inhibitor)
- CAS:
- MF:
- Chemical Name:NU-7441 (DNA-PK inhibitor)
- CAS:
- MF:
- Chemical Name:MG-132 (PROTEASOME Inhibitor)
- CAS:
- MF:
- Chemical Name:MASITINIB (C-KIT inhibitor)
- CAS:
- MF:
- Chemical Name:IXAZEOMIB (MLN2238) (20S PROTEASOME Inhibitor)
- CAS:
- MF:
- Chemical Name:ICOTINIB HCL (EGFR inhibitor)
- CAS:
- MF:
- Structure:

- Chemical Name:HYDROXYLAMINE HYDROCHLORIDE/Hydroxylamine Hydrochloride
- CAS:
- MF:Cl2H8N2O2
- Chemical Name:EPOTHILONE B (MICROTUBULE ASSOSIATED inhibitor)
- CAS:
- MF:
- Chemical Name:WH-4-023 (SRC inhibitor)
- CAS:
- MF:
- Chemical Name:TG101348 (JAK inhibitor)
- CAS:
- MF:
- Chemical Name:PFI-3 (EPIGENETIC READER DOMAIN inhibitor)
- CAS:
- MF:
- Chemical Name:PD184352 (MEK inhibitor)
- CAS:
- MF:
- Chemical Name:ML324 (HISTONE DEMETHYLASE inhibitor)
- CAS:
- MF:
- Chemical Name:KU0063794 (MTOR inhibitor)
- CAS:
- MF:
- Chemical Name:JNJ-7777120 (HISTAMINE RECEPTOR antagonist)
- CAS:
- MF:
- Chemical Name:GSK1292263 (GPR agonist)
- CAS:
- MF:
- Chemical Name:BYL719 (PI3K inhibitor)
- CAS:
- MF:
- Chemical Name:BML-210 (HDAC inhibitor)
- CAS:
- MF:
- Structure:

- Chemical Name:2H-Pyran-4-propanamide, α-[4-(cyclopropylsulfonyl)phenyl]-N-(5-fluoro-2-thiazolyl)tetrahydro-, (αR)-
- CAS:745051-61-0
- MF:C20H23FN2O4S2
- Chemical Name:VENETOCLAX (ABT-199, GDC-0199) (BCL-2 inhibitor)
- CAS:
- MF:
- Chemical Name:U-104 (Carbonic anhydrase inhibitor)
- CAS:
- MF:
- Chemical Name:E-64 (CYSTEINE PROTEASE inhibitor)
- CAS:
- MF:
- Chemical Name:DOCETAXEL (MICROTUBULE ASSOSIATED inhibitor)
- CAS:
- MF:
- Chemical Name:DEGRASYN (BCR-ABL inhibitor)
- CAS:
- MF:
- Chemical Name:CC-223 (MTOR inhibitor)
- CAS:
- MF:
- Chemical Name:BI2536 (PLK inhibitor)
- CAS:
- MF:
- Chemical Name:A83-01 (ALK5 inhibitor)
- CAS:
- MF:
- Chemical Name:A-366 (HISTONE METHYLTRANSFERASE Inhibitor)
- CAS:
- MF:
- Structure:

- Chemical Name:ICA 069673
- CAS:582323-16-8
- MF:C11H6ClF2N3O
- Chemical Name:VOLASERTIB (PLK inhibitor)
- CAS:
- MF:
- Chemical Name:TUBASTATIN A (HDAC inhibitor)
- CAS:
- MF:
- Chemical Name:TEDIZOLID (MAO-A inhibitor)
- CAS:
- MF:
- Chemical Name:SP600125 (JNK inhibitor)
- CAS:
- MF:
- Chemical Name:SB203580 (P38 MAPK Inhibitor)
- CAS:
- MF:
- Chemical Name:SALIRASIB (RHO inhibitor)
- CAS:
- MF:
- Chemical Name:RG108 (DNA METHYLTRANSFERASE inhibitor)
- CAS:
- MF:
- Chemical Name:PLERIXAFOR (CXCR inhibitor)
- CAS:
- MF:
- Chemical Name:PD-173955 (BCR-ABL inhibitor)
- CAS:
- MF:
- Chemical Name:ODANACATIB (CYSTEINE PROTEASE inhibitor)
- CAS:
- MF:
- Chemical Name:MI-2 (HISTONE METHYLTRANSFERASE Inhibitor)
- CAS:
- MF:
- Chemical Name:GSK1278863 (HIF inhibitor)
- CAS:
- MF:
- Chemical Name:DACOMITINIB (EGFR inhibitor)
- CAS:
- MF:
- Chemical Name:BATIMASTAT (MMP inhibitor)
- CAS:
- MF:
- Chemical Name:AVASIMIBE (P450 inhibitor)
- CAS:
- MF:
- Chemical Name:SALUBRINAL (PERK inhibitor)
- CAS:
- MF:
- Chemical Name:FLAVOPIRIDOL HCL (CDK inhibitor)
- CAS:
- MF:
- Chemical Name:DEFACTINIB (FAK inhibitor)
- CAS:
- MF:
- Chemical Name:CEDIRANIB (VEGFR inhibitor)
- CAS:
- MF:
- Chemical Name:BAY11-7082 (IΚB/IKK inhibitor)
- CAS:
- MF:
- Chemical Name:(-)-BLEBBISTATIN (ATPASE inhibitor)
- CAS:
- MF:
- Chemical Name:AG14361 (PARP1 inhibitor)
- CAS:
- MF:
- Chemical Name:ACP-196 (BTK inhibitor)
- CAS:
- MF:
- Chemical Name:ABT-737 (BCL-2 inhibitor)
- CAS:
- MF:
- Structure:

- Chemical Name:CK-2127107
- CAS:1345410-31-2
- MF:C19H18F2N6O
- Chemical Name:VILAZODONE (SSRI inhibitor)
- CAS:
- MF:
- Chemical Name:TBA-354 (anti-tuberculosis)
- CAS:
- MF:
- Chemical Name:SAG (HEDGEHOG/SMOOTHENED agonist)
- CAS:
- MF:
- Chemical Name:PACLITAXEL (MICROTUBULE ASSOSIATED inhibitor)
- CAS:
- MF:
- Chemical Name:OSU-03012 (PDK-1 inhibitor)
- CAS:
- MF:
- Chemical Name:MONOMETHYL AURISTATIN E (microtubule-associated inhibitor)
- CAS:
- MF:
- Chemical Name:ML141 (RHO inhibitor)
- CAS:
- MF:
- Chemical Name:KN-93 PHOSPHATE (CAMK Inhibitor)
- CAS:
- MF:
- Chemical Name:GSK126 (EZH2 inhibitor)
- CAS:
- MF:
- Chemical Name:GELDANAMYCIN (HSP90 inhibitor)
- CAS:
- MF:
- Chemical Name:GANT61 (HEDGEHOG/SMOOTHENED Inhibitor)
- CAS:
- MF:
- Chemical Name:EPZ-6438 (E7438) (EZH2 inhibitor)
- CAS:
- MF:
- Chemical Name:EMPAGLIFLOZIN (SGLT inhibitor)
- CAS:
- MF:
- Chemical Name:DOXORUBICIN (TOPOISOMERASE inhibitor)
- CAS:
- MF:
- Chemical Name:DAPT (Γ-SECRETASE inhibitor)
- CAS:
- MF:
- Chemical Name:DACLATASVIR (HCV NS5A inhibitor)
- CAS:
- MF:
- Chemical Name:COMBRETASTATIN A4 (MICROTUBULE ASSOCIATED inhibitor)
- CAS:
- MF:
- Chemical Name:CABOZANTINIB (VEGFR inhibitor)
- CAS:
- MF:
- Chemical Name:BREFELDIN A (protein transport inhibitor)
- CAS:
- MF:
- Chemical Name:BKM120 (PI3K inhibitor)
- CAS:
- MF:
- Chemical Name:AKT INHIBITOR VIII (AKT inhibitor)
- CAS:
- MF:
- Chemical Name:ABT-199 (BCL-2 inhibitor)
- CAS:
- MF:
- Structure:

- Chemical Name:Porfiromycin
- CAS:801-52-5
- MF:C16H20N4O5
- Chemical Name:VINCRISTINE (MICROTUBULE ASSOSIATED inhibitor)
- CAS:
- MF:
- Chemical Name:TETRABENAZINE (VMAT-2 Inhibitor)
- CAS:
- MF:
- Chemical Name:SNX-2112 (PF-04928473) (HSP90 antimony inhibitor)
- CAS:
- MF:
- Chemical Name:PLX4032 (RAF inhibitor)
- CAS:
- MF:
- Chemical Name:PD123319 (RAAS inhibitor)
- CAS:
- MF:
- Chemical Name:NS-2028 (SGC inhibitor)
- CAS:
- MF:
- Chemical Name:NECROSTATIN-1 (TNF-ALPHA inhibitor)
- CAS:
- MF:
- Chemical Name:ML323 (DUB inhibitor)
- CAS:
- MF:
- Chemical Name:KU-55933 (ATM inhibitor)
- CAS:
- MF:
- Chemical Name:(+)-JQ1 (BRD4 inhibitor)
- CAS:
- MF:
- Chemical Name:GSK2141795 (AKT inhibitor)
- CAS:
- MF:
- Chemical Name:GANETESPIB (HSP inhibitor)
- CAS:
- MF:
- Chemical Name:ENZALUTAMIDE (MDV3100) (AR inhibitor)
- CAS:
- MF: