3-[(2-Methyl-1,3-thiazol-4-yl)ethynyl]pyridine hydrochloride Chemical Properties,Usage,Production
Biological Activity
Potent, selective and non-competitive mGlu 5 antagonist (IC 50 = 5 nM in Ca 2+ -flux assay; K i = 16 nM). Displays anxiolytic activity in vivo and is orally active.