BISINDOLYLMALEIMIDE X HYDROCHLORIDE (BIM-X HYDROCHLORIDE)

生物活性靶点体外研究

CAS号:145317-11-9
英文名:1H-Pyrrole-2,5-dione, 3-[8-(aMinoMethyl)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl]-4-(1-Methyl-1H-indol-3-yl)-, Monohy
中文名:BISINDOLYLMALEIMIDE X HYDROCHLORIDE (BIM-X HYDROCHLORIDE)
CBNumber:CB82667395
分子式:C26H25ClN4O2
分子量:460.96
MOL File:145317-11-9.mol

BISINDOLYLMALEIMIDE X HYDROCHLORIDE (BIM-X HYDROCHLORIDE)化学性质

储存条件 :under inert gas (nitrogen or Argon) at 2-8°C
溶解度 :Soluble in DMSO (up to 10 mg/ml)
形态 :Red solid.
颜色 :Red
生物来源 :synthetic (organic)
稳定性 :Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.

BISINDOLYLMALEIMIDE X HYDROCHLORIDE (BIM-X HYDROCHLORIDE)性质、用途与生产工艺

生物活性 Bisindolylmaleimide X hydrochloride (BIM-X hydrochloride) 是一种有效的，选择性的蛋白激酶 C (PKC) 抑制剂。Bisindolylmaleimide X hydrochloride 也是一种有效的细胞周期蛋白依赖性激酶 2 (CDK2) 拮抗剂，IC50 为 200 nM。
靶点

CDK2

200 nM (IC ₅₀ )

PKC
体外研究

Bisindolylmaleimide X hydrochloride (BIM-X hydrochloride; Ro31-8425 hydrochloride) derivatives acts as an useful tool to compare inhibitor potencies and selectivities for a target of interest.

BISINDOLYLMALEIMIDE X HYDROCHLORIDE (BIM-X HYDROCHLORIDE)上下游产品信息

上游原料

下游产品

BISINDOLYLMALEIMIDE X HYDROCHLORIDE (BIM-X HYDROCHLORIDE)生产厂家

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