生物活性 靶点 体外研究
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AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE

AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE,167114-91-2,结构式
AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE
  • CAS号:167114-91-2
  • 英文名:AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE
  • 中文名:AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE
  • CBNumber:CB7671283
  • 分子式:C64H116N22O19
  • 分子量:1497.74
  • MOL File:167114-91-2.mol
AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE化学性质
  • 储存条件 :-20°C
  • 溶解度 :H2O: soluble
  • 形态 :lyophilized powder
  • 颜色 :white
  • 水溶解性 :Soluble to 1 mg/ml in water
安全信息

AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE性质、用途与生产工艺

  • 生物活性 Autocamtide-2-related inhibitory peptide 是高度特异性的、CaMKII 的有效抑制剂,其IC50 值为 40 nM。
  • 靶点

    IC50: 40 nM (CaMKII).

  • 体外研究

    It is found that Autocamtide-2-related inhibitory peptide (a novel synthetic peptide ATP) is a potent inhibitor of CaM-kinase II with an IC 50 of 40 nM, which is active in the presence or absence of Ca 2+ /calmodulin. It is 50 and 500 times more potent than CaMK-(281-302Ala286) and KN-93,respectively, under the assay condition used.

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AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE生产厂家
  • 公司名称:Carbosynth
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