105277-43-8
中文名称
PD 119819
英文名称
PD 119819
CAS
105277-43-8
分子式
C21H24ClN3O3
分子量
401.89
MOL 文件
105277-43-8.mol
结构式
基本信息
中文别名
化合物 T28318
英文别名
PD 119819
PD119819' PD-119819
7-<3-<4-(2-pyridinyl)-1-piperazinyl>propoxy>-4H-1-benzopyran-4-one dihydrochloride
PD119819' PD-119819
7-<3-<4-(2-pyridinyl)-1-piperazinyl>propoxy>-4H-1-benzopyran-4-one dihydrochloride
应用领域
用途一
PD 119819 is a heterocyclic piperazine and has been identified as an extremely selective DA autoreceptor agonist in tests that include [3H]haloperidol binding, inhibition of spontaneous locomotor activity, inhibition of brain DA synthesis, inhibition of brain DA neuronal firing, stereotypy assessment, and reversal of 6-hydroxydopamine (6-OHDA) induced akinesia in rats.
常见问题列表
概述
PD 119819 是一种高选择性 benzopyran-4-one brain dopamine autoreceptor 激动剂。PD 119819 是一种杂环哌嗪,可抑制自发运动活动和脑 dopamine 合成。