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4-Iodobut-1-ene is a reagent in the design of cell-permeable stapled peptides which are used as HIV-1 integrase inhibitors. 4-Iodobut-1-ene is also used as a reagent in the synthesis of pyrrolopyridazines as novel DGAT1 inhibitors.

Tetrahedron Letters, 31, p. 937, 1990 DOI: 10.1016/S0040-4039(00)94397-1