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Crotonyl fentanyl is an analytical reference material categorized as an opioid.^1,2,3 Crotonyl fentanyl induces generalized responses in mice trained to discriminate oxycodone from saline.⁴ Crotonyl fentanyl is regulated as a Schedule I compound in the United States. This product is intended for research and forensic applications.

Crotonyl Fentanyl is an analog of Fentanyl (F274990), which is a controlled substanced used as analgesic.

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2. Vasudevan, L., Vandeputte, M.M., Deventer, M., et al. Assessment of structure-activity relationships and biased agonism at the mu opioid receptor of novel synthetic opioids using a novel, stable bio-assay platform Biochem. Pharmacol. 177,113910(2020).
3. Varshneya, N.B., Walentiny, D.M., Moisa, L.T., et al. Opioid-like antinociceptive and locomotor effects of emerging fentanyl-related substances Neuropharmacology 151,171-179(2019).
4. Walentiny, D.M., Moisa, L.T., and Beardsley, P.M. Oxycodone-like discriminative stimulus effects of fentanyl-related emerging drugs of abuse in mice Neuropharmacology 150,210-216(2019).