RXFP1 receptor agonist-5 (Example 98) is a RXFP1 receptor agonist. RXFP1 receptor agonist-5 stimulates cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 1.3 nM[1].
References
[1] Sreekantha Ratna KUMAR, et al. Benzothiazole, benzoisoxazole and benzodioxole analogs as rxfp1 receptor agonists. Patent. WO2023114822A1.
