RXFP1 receptor agonist-2 (Example 124) is a RXFP1 receptor agonist. RXFP1 receptor agonist-2 stimulates cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 1 nM[1].
References
[1] Scott A. SHAW, et al. Rxfp1 agonists. Patent. WO2023077040.
