NSD2-PWWP1-IN-2 (compound 33) is a potent NSD2-PWWP1 inhibitor with an IC50 value of 1.49 μM. NSD2-PWWP1-IN-2 has the potential for the research of cancer[1].
IC 50
NSD2: 1.49 μM (IC50)
References
[1] Li N, et al. Structure-Based Discovery of a Series of NSD2-PWWP1 Inhibitors. J Med Chem. 2022 Jul 14;65(13):9459-9477. DOI:10.1021/acs.jmedchem.2c00709
