2624313-15-9

dTAGV-1 (35 mg/kg; i.p. once daily for 4 days) TFA induces degradation of FKBP12^F36V-Nluc in mice^[1].
dTAGV-1 (2-10 mg/kg; i.p.) TFA exhbits half-lives (T_1/2=3.64 and 4.4 h), C_max (595 and 2123 ng/mL) and great exposure (AUC_inf?=3136 and?18517 h?ng/mL) in mice^[1].
dTAGV-1 (2 mg/kg; i.v.) TFA exhbits half-life (T_1/2=3.02 h), C_max (7780 ng/mL) and great exposure (AUC_inf?=3329 h?ng/mL) in mice^[1].