192053-05-7

MRS 1334 is a potent and highly selective hA3 antagonist.

ChEBI: 2-methyl-6-phenyl-4-(2-phenylethynyl)-1,4-dihydropyridine-3,5-dicarboxylic acid O3-ethyl ester O5-[(4-nitrophenyl)methyl] ester is a cinnamate ester.

Potent and highly selective antagonist for the human adenosine A 3 receptor. K i values are 2.69 nM at hA 3 , and > 100 μ M at rat A 1 and rat A 2A receptors.

hA₃: 2.69 nM (Ki); rA₁: >100 nM (Ki); rA_2A: >100 nM (Ki)

Desiccate at -20°C