186002-54-0

.alpha.2A-Adrenoceptor antagonism increases insulin secretion and synergistically augments insulinotropic effect of glibenclamide.

rat α2A receptor: 0.42 nM (Kd); rat α2B recepter: 0.18 nM (Kd); rat α2C recepter: 0.19 nM (Kd); human α2A-adrenoceptor: 0.6 nM (Kd); human α2B-adrenoceptor: 0.46 nM (Kd); human α2C-adrenoceptor: 0.77 nM (Kd)

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