176199-48-7

Treatment ofgeneral anxiety disorders and smoking cessation (metabotropic glutamate agonist).

ChEBI: Eglumetad is a L-alpha-amino acid.

Highly selective and potent agonist of group II mGlu receptors (EC 50 values are 5.1 and 24.3 nM at mGlu 2 and mGlu 3 receptors respectively and > 100000 nM at mGlu 4 , mGlu 7 , mGlu 1a and mGlu 5a receptors). Displays antianxiety and antiaddictive activity in vivo . Orally and systemically active.

+4°C