1427521-34-3

AM2201 is a potent synthetic cannabinoid (CB) with K_i values of 1.0 and 2.6 nM for the CB₁ and CB₂ receptors, respectively.¹ AM2201 N-(4-hydroxypentyl) metabolite is an expected urinary metabolite of AM2201, based on the known metabolism of similar compounds.² Its biological actions are unknown.

4-Hydroxypentyl AM-2201 is a metabolite of AM-2201 (A575830), is a drug which acts as a potent but unselective agonist for the cannabinoid receptor CB1 or CB2.

1. Makriyannis, A., and Deng, H. Cannabimimetic indole derivatives US7241799B2,(2001).
2. Wintermeyer, A., M?ller, I., Thevis, M., et al. In vitro phase I metabolism of the synthetic cannabimimetic JWH-018 Anal. Bioanal. Chem. 398(5),2141-2153(2010).