141064-23-5

Muscarinic receptors are G protein-coupled acetylcholine receptors that play diverse roles. Xanomeline (oxalate) is a potent agonist of muscarinic acetylcholine receptors (EC₅₀ values are 0.3, 92.5, 5, 52, and 42 nM for M₁, M₂, M₃, M₄, and M₅, respectively). It has antipsychotic-like activities in rats and Cebus monkeys. M₁ selective agonists, like Xanomeline (oxalate), enhance memory function and has utility in treating Alzheimer’s Disease.

Xanomeline oxalate is a functionally selective mAChR M1 agonist.

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