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MEN 10207 is a tachykinin antagonist.

MEN 10207 is a selective NK-2 tachykinin receptor (Neurokinin Receptor) antagonist. MEN 10207 has pA2 values of 5.2, 7.9 and 4.9 in three monoreceptor in vitro assays for NK-1, NK-2 and NK-3 tachykinin receptors, respectively.

Tachykinin NK₂ Receptor: 7.9 (pA2); NK1: 5.2 (pA2); NK3: 4.9 (pA2)

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