5-chloro-3-ethyl-1H-indole-2-carboxylic acid [2-(4-piperidin-1-yl-phenyl)-ethyl]-amide
- русский язык имя
- английское имя5-chloro-3-ethyl-1H-indole-2-carboxylic acid [2-(4-piperidin-1-yl-phenyl)-ethyl]-amide
- CAS №868273-06-7
- CBNumberCB42092872
- ФормулаC24H28ClN3O
- мольный вес409.95
- EINECS278-169-7
- номер MDLMFCD11045300
- файл Mol868273-06-7.mol
химическое свойство
| Температура кипения | 660.3±55.0 °C(Predicted) |
| плотность | 1.218±0.06 g/cm3(Predicted) |
| температура хранения | 2-8°C |
| растворимость | H2O: <2mg/mL |
| форма | powder |
| пка | 14.87±0.30(Predicted) |
| цвет | white |
| FDA UNII | 7YW2S3Z2CB |
5-chloro-3-ethyl-1H-indole-2-carboxylic acid [2-(4-piperidin-1-yl-phenyl)-ethyl]-amide химические свойства, назначение, производство
Использование
Org 27569 is a drug that is a used in biological studies for structure-activity relationships of indole-carboxamides as CB1 receptor allosteric modulators.Биологическая активность
Potent CB 1 receptor allosteric modulator (pEC 50 = 8.24). Significantly increases binding of the CB 1 agonist [ 3 H]CP 55.940 (pK b = 5.67) and decreases binding of the CB 1 inverse agonist [ 3 H]SR 141716A (pK b = 5.95). Inhibits CB 1 receptor antagonist efficacy in vitro (pK b = 7.57).5-chloro-3-ethyl-1H-indole-2-carboxylic acid [2-(4-piperidin-1-yl-phenyl)-ethyl]-amide поставщик
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