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  • VGSC blocker-1|T39717|TargetMol

VGSC blocker-1|T39717|TargetMol

VGSC blocker-1
￥10600 25mg 起订
￥17500 100mg 起订
￥13800 50mg 起订
上海 更新日期：2026-05-09

TargetMol 中国（陶术生物）

VIP1年
联系人：邵经理
电话：400-821-0310拨打
手机：15002144251 拨打
邮箱：xuexiang.shao@tsbiochem.com

产品详情:

中文名称：
VGSC blocker-1
英文名称：
VGSC blocker-1
CAS号：
2230472-55-4
品牌：
TargetMol
产地：
美国
保存条件：
Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature.
产品类别：
抑制剂
货号：
T39717

Product Introduction

Bioactivity

名称VGSC blocker-1
描述VGSC blocker-1 is a powerful small molecule that serves as a blocker for the neonatal isoform of the VGSC subtype known as Nav1.5 (nNav1.5). It effectively blocks INa peak currents by 34.9% at a concentration of 1 μM, and demonstrates a 0.3% inhibition of cell invasion at the same concentration in the MDA-MB-231 human breast cancer cell line, without compromising cell viability.
体外活性VGSC blocker 1 (compound 1) (1.0 to 10 μM) inhibits human breast cancer cell line MDA-MB-231[1]. Cell Viability Assay[1]Cell Line: human breast cancer cell line MDA-MB-231 Concentration: 1.0 to 10μM Incubation Time: 24 hours Result: VGSC blocker 1 blocks INa peak currents 34.9% at 1 uMa and inhibits cell invasion 0.3% at 1 uM. These values are much higher than the concentrations required (0.1 μM and 1 μM) to produce significant nNav1.5 current blockade and cell invasion inhibition.
存储条件Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature.
关键字VGSC blocker-1 | VGSC blocker1 | VGSC blocker 1
相关产品Lidocaine hydrochloride | Dibucaine | Valproic Acid | Lidocaine | Mebeverine hydrochloride | Safinamide | Procaine | L-Aspartic aicd sodium | Permethrin | Tetracaine hydrochloride | Phenytoin sodium | Ranolazine dihydrochloride
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VGSC blocker-1|TargetMol

公司简介


成立日期 (14年)
注册资本 589.8595万人民币
员工人数 100-500人
年营业额 ￥ 1亿以上
经营模式 贸易,工厂,试剂,定制,服务
主营行业 天然产物,生物化工,化学试剂,生物技术服务

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