| Name | Litorin acetate(55749-97-8 Free base) |
| Description | Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist. It stimulates the contraction of smooth muscle, stimulates gastrin, gastric acid, and pancreatic secretion, and suppresses the nutriment in vivo. |
| In vitro | 99mTc-Litorin is developed for non-invasive imaging of tumors with overexpressed gastrin-releasing peptide receptors (GRP-R)[1].
[D-Phe1,Leu8,9]Litorin inhibits binding of 125I-[Tyr4] BN to murine Swiss 3T3 cells with a Ki of 5.1 nM[2].
Litorin stimulates 3H-Thymidine incorporation in murine Swiss 3T3 cells with an EC50 of 2.3 nM[2]. |
| In vivo | Litorin stimulates the contraction of smooth muscle, stimulates gastrin, gastric acid, and pancreatic secretion, and suppresses the nutriment in in vivo experiments[2]. |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| Keywords | Litorin acetate | Litorin acetate(55749-97-8 Free base) |
| Inhibitors Related | [D-Phe12]-Bombesin acetate | BA 1 acetate(183241-31-8 free base) | MK-5046 | [D-Phe12,Leu14]-Bombesin acetate | ML-18 | Bombesin acetate(31362-50-2 free base) | kuwanon G | Kuwanon H | CD80-IN-3 | PD176252 |
| Related Compound Libraries | Bioactive Compound Library | Membrane Protein-targeted Compound Library | Natural Product Library | Peptide Compound Library | Natural Product Library for HTS | Bioactive Compounds Library Max | GPCR Compound Library |
United States
