BRL 50481

▼

▲

Product Name:

BRL 50481

Synonyms:

5-NITRO-2,N,N-TRIMETHYLBENZENESULFONAMIDE;BRL 50481;N,N,2-TRIMETHYL-5-NITRO-BENZENESULFONAMIDE;3-(N,N-Dimethylsulfonamido)-4-methylnitrobenzene,5-Nitro-2-N,N-trimethylbenzenesulfonamide;Benzenesulfonamide, N,N,2-trimethyl-5-nitro-

CAS:

433695-36-4

MF:

C9H12N2O4S

MW:

244.27

EINECS:

1592732-453-0

Product Categories:

All Inhibitors;Inhibitors;Cyclic Nucleotide related

Mol File:

433695-36-4.mol

▼

▲

BRL 50481 Chemical Properties

▼

▲

Melting point

65-67°C

Boiling point

391.1±52.0 °C(Predicted)

density

1.334±0.06 g/cm3(Predicted)

storage temp.

2-8°C

solubility

DMSO: 12 mg/mL

pka

-5?+-.0.70(Predicted)

form

solid

color

white

▼

▲

BRL 50481 Usage And Synthesis

▼

▲

Chemical Properties

Off-White Solid

Uses

A PDE7 inhibitor that has acceptable selectivity for in vivo studies

Biological Activity

Selective, substrate-competitive inhibitor of phosphodiesterase (PDE) 7 (K i = 180 nM). Displays > 200-fold selectivity over PDE1B, PDE1C, PDE2, PDE3, PDE4A4 and PDE5.

Product Name	BRL 50481
CAS No	433695-36-4
EC-No
Min. Order	1g
Purity	99%
Supply Ability	200kg
Release date	2019/12/27

Company Profile Introduction

You may like

Recommended supplier