Tianeptine Sulfate
Other name: Tianeptine hemisulfate monohydrate
CAS : 1224690-84-9
Mol. Formula: C21H27ClN2O8S2
Tianeptine Sulfate/Tianeptine hemisulfate monohydrate is an improved salt of Tianeptine. It is not hygroscopic so handling the powder is a lot easier. Since it is not as readily absorbed and excreted from the body, the sulfate salt allows for a more controlled release of the Tianeptine over longer periods. Rather than having to dose three times with rapid peak effects and rapidly falling effects, the sulfate salt allows for one dose to maintain plasma levels in the body much longer than the sodium salt. These improved characteristics make Tianeptine Sulfate a novel addition.
Function
Tianeptine Sulfate not only a good antidepressant effect and adverse reactions was significantly less than conventional antidepressant tricyclic drugs, almost no adverse effect on the cardiovascular system, blood , liver and kidney functions were not hurt, nor do I have a calming effect. Tianeptine is not only effective for depression and depressive neurosis, chronic alcoholism and depression after alcohol is also effective. Long-term use can prevent relapse
Specification
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Items
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Specifications
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Results
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Appearance
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White crystalline powder
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Complies
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Solubility
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Soluble in dimethylformamide,insoluble in water and dichloromethane
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Complies
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Impurity A
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≤0.1%
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Not detected
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Identification
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Infrared spectrum should be consistent with the reference spectra
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Complies
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Should show the identification of sulfate reaction
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Complies
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Water
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≤5.0%
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3.85%
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Organic residues
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Ethyl acetate≤0.5%
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Not detected
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Dichloromethane≤0.06%
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Not detected
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Methanol≤0.3%
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Not detected
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Acetone≤0.5%
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Not detected
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Acetonitrile≤0.041%
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Nor detected
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Ethanol≤0.5%
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0.099%
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N,N-dimethyiformamide≤0.088%
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Nor detected
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Assay
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99.0%-101.0%
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99.57%
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China
