Nice Price Tianeptine Sodium Salt Powder 99% 30123-17-2 Tianeptine Sodium
Product discription
Product Name: | Tianeptine sodium salt |
Synonyms: | TIANEPTINE SODIUM;TIANEPTINE SODIUM SALT;7-[(3-Chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic Acid S,S-Dioxide Sodium Salt;S-1574;Stablon;7-[(3-chloro-6,11-dihydro-6-methyl-dibenzo[c,f][1,2]thiazepine-11-yl)amino]heptanoic acid s,s dioxide sodium salt;[7-[(3-Chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepine 5,5-dioxide)-11-ylamino]heptanoic acid]sodium salt;3-Chloro-6,11-dihydro-6-methyl-11-[6-(sodiooxycarbonyl)hexylamino]dibenzo[c,f][1,2]thiazepine 5,5-dioxide |
CAS: | 30123-17-2 |
MF: | C21H24ClN2NaO4S |
MW: | 458.93 |
EINECS: | 250-059-3 |
Product Categories: | chemical;Stablon, Coaxil, Tatinol;Intermediates & Fine Chemicals;Pharmaceuticals;API;Inhibitors;Heterocycles;Sulfur & Selenium Compounds;Tianeptine sodi |
Mol File: | 30123-17-2.mol |
Tianeptine sodium salt is a salt of Tianeptine. Tianeptine is an atypical antidepressant. It is an agonist of the μ-opioid receptor (MOR; EC50s = 194 and 641 nM for human and mouse receptors, respectively, in a BRET assay for G protein activation) and also has effects on the glutamate system. Tianeptine (30 mg/kg) decreases immobility in the forced swim test in wild-type, but not MOR knockout mice, indicating antidepressant-like activity dependent on MORs. It increases locomotor activity at a dose of 30, but not 10 mg/kg, in the open field test and increases paw withdrawal latency in the hot-plate test in mice. Tianeptine modulates AMPA receptor activity by increasing phosphorylation of the AMPA receptor GluR1 subunit in the frontal cortex and hippocampal CA3 region in mice. It prevents increases in glial glutamate transporter 1 (GLT-1) expression induced by chronic restraint stress in the hippocampal CA3 region in rats when administered at a dose of 10 mg/kg per day for 21 days.5It also reverses increases in extracellular glutamate levels induced by acute restraint stress in the basolateral nucleus of the amygdala in rats.
Usage And Synthesis
Tianeptine Sodium Salt is a tricyclic compound with psychostimulant, anti-ulcer and anti-emetic properties. Antidepressant.
Tianeptine sodium salt hydrate has been used as a selective serotonin reuptake enhancer (SSRE) positive control during serotonin transporter (SERT) assay in human embryonic kidney 293 cell lines.
Tricyclic compound with psychostimulant, anti-ulcer and anti-emetic properties. Antidepressant.
Our Service
1.Cooperate with research institutions, we strictly control the process from raw material to finished product.
2.We can provide the reasonable price, high quality products and prompt shipment.
3.We can send the goods to your delivery address directly. It is relatively safe and fast.
4.Quick and clear response to customers questions, we’ll treat every email and message within 24 hours usually much faster.
5.We can provide you a discount if you place a substantial order with us.
6.Products can be packaged and company logo can be customized according to customer requirements.
Our company
Guangzhou Biocar Biotechnology Co.,Ltd.,formerly known as Guangdong Yangye Pharmaceutical Factory established in 2005, which is affiliated to Wuhan Biocar Group. With the rise of Internet +, company's business process is accelerating. The company's board of directors has decided to establish Guangzhou Yangye Biotechnology Co., Ltd. at the end of 2016.
Guangzhou Biocar Biotechnology Co.,Ltd. is located near Zhujiang New Town, Tianhe District, one of the prosperous areas in Guangzhou. This helps facilitate business negotiations at home and abroad. It is a high-tech enterprise centered in Guangdong, radiating across our country and facing the world. And it is mainly engaged in the research, development and sales of new chemical raw materials, the custom synthesis and import and export of pharmaceutical intermediates and APIs, the agency sales of pharmaceutical chemicals, the research and development, production and sales of flavors, fragrances and chemical raw materials. Its factory covers an area of more than 4,000 acres and has more than 600 employees.
Guangzhou Biocar Biotechnology has a production base for deep processing of feed additives and veterinary drug intermediates based on main pharmaceutical intermediates.
It has always adhered to the tenet of "Being faithful, cultivating harmony and achieving win-win cooperation" and treats every customer sincerely.
We are looking forward to cooperating with you sincerely, and making mutual benefit and brilliance!
Delivery
1. Sent out in 24hours once payment comfirm.
2. Professional agent make sure our ship fastly and safety
3.Offer your tracking number to you once we get it ,in order to facilitateyou track the express
FAQ
Q1: Can i get some samples?
A: Yes, we can supply the sample, but the shipping cost be paid by ourcustomers.
Q2: How to start orders or make payments?
A: Proforma invoice will be sent first after confirmation of order, enclosedour bank information. Payment by T/T, Western Union or Paypal.
Q3: How to confirm the Product Quality before placing orders?
A:You can get free samples for some products,you only need to pay theshipping cost or arrange a courier to us and take the samples. You cansend us your product specifications and requests,we will manufacture theproducts according to your requests.
Q4:What's your MOQ?
A:Our MOQ is 1kg. But usually we accept less quantity such as 100g onthe condition that sample charge is 100% paid.
Q5: How about delivery lead time?
A:Delivery lead time: About 3-5 days after payment confirmed. (Chineseholiday not included)
Q6: Do You Ship Over The Weekend?
We use EMS,TNT,FEDEX,DHL four kinds of couriers. EMS don't collected parcelsover the weekend. The packages can be shipped out normally before 12:00a.m in Beijing time if you choose to ship by TNT or FedEx.
Transaction requirements: serious and sincere, pragmatic and efficient
1. We support the verification of the authenticity of our warehouse andproducts through video conversations.
2. If we release this product, it means that we can also produce its similarproducts.
3. We have insured each product, if the goods are lost or damaged, wecan provide a 100% refund.
4. Delivery time limit: 4-7 days in the UK, 10-15 days in other countries.
5. Company qualification: Seven years since its establishment, with 2factories and 8 laboratories,has cooperated with Wuhan Textile Universityand set up a talent reserve base, which can accept the customization ofpharmaceutical intermediates and the mass production of large chemicals.
6. Quality inspection certificate: every product has its third-party qualityinspection certificate to ensure the safety of the product.
7. Advantages: can be customized production, can be shipped in batches,price concessions, high timeliness.
8.Can assist customers in brand design and printing, and has successfullybuilt OMEGA, ZE and other brands
9. Payment method: Western Union, MoneyGram, Bitcoin, bank transfer, remitlyare currently accepted.
10.Reject malicious inquiries, reject scammers
11.Provide door-to-door transportation, as well as normal customs clearanceservices