2-(3-羧基丙基)-3-氨基-6-(4-甲氧苯基)吡啶溴化
2-(3-羧基丙基)-3-氨基-6-(4-甲氧苯基)吡啶溴化
2-(3-羧基丙基)-3-氨基-6-(4-甲氧苯基)吡啶溴化 性质
| 熔点 | 200 °C(Solv: ethanol (64-17-5)) |
|---|---|
| 储存条件 | Store at RT |
| 溶解度 | 在DMSO中的溶解度为30 毫克/毫升 |
| 形态 | 固体 |
| 颜色 | 白色 |
| 水溶解性 | water: 25mM |
| InChI | 1S/C15H17N3O3.BrH/c1-21-12-6-4-11(5-7-12)13-8-9-14(16)18(17-13)10-2-3-15(19)20;/h4-9,16H,2-3,10H2,1H3,(H,19,20);1H |
| InChIKey | GFZHNFOGCMEYTA-UHFFFAOYSA-N |
| SMILES | [Br-].COc1ccc(cc1)-c2ccc(N)[n+](CCCC(O)=O)n2 |
2-(3-羧基丙基)-3-氨基-6-(4-甲氧苯基)吡啶溴化 用途与合成方法
0.2 μM (GABA receptor).
Both bicuculline and Gabazine (SR 95531) have been characterized as competitive inhibitors of GABA binding to the GABA A receptor. Gabazine is more potent than bicuculline at blocking currents elicited by GABA, with an IC 50 for currents elicited by 3 μM GABA of ~0.2 μM and a Hill coefficient of 1.0. Gabazine reduces the currents elicited by 10 μM alphaxalone by ~30%, for responses of receptors containing wildtype β2 subunits. The concentration of Gabazine requires producing half the maximal block is ~0.2 μM. Gabazine also could only produce a partial block of currents gated by 300 μM pentobarbital. The maximal reduction, again, is ~30%, and the concentration of Gabazine required to produce half the maximal block is ~0.15 μM.
2-(3-羧基丙基)-3-氨基-6-(4-甲氧苯基)吡啶溴化 价格(试剂级)
| 更新日期 | 产品编号 | 产品名称 | CAS号 | 包装 | 价格 |
|---|---|---|---|---|---|
| 2026-06-05 | HY-103533R | 2-(3-羧基丙基)-3-氨基-6-(4-甲氧苯基)吡啶溴化 | 104104-50-9 | 5 mg | 1400 |
| 2026-06-05 | HY-103533 | 2-(3-羧基丙基)-3-氨基-6-(4-甲氧苯基)吡啶溴化 | 104104-50-9 | 1 mg | 272 |
