Phenol, 2-methoxy-4-[3-(phenylamino)imidazo[1,2-a]pyrazin-2-yl]-

SDR-04 is a?BET?inhibitor and exhibits strong BRD4-BD1 affinity and inhibition activity. SDR-04 potently suppresses MV4;11 cancer cell line proliferation[1].

BD1

[1] Ru Dong, et al. Design, synthesis and anticancer evaluation of 3-methyl-1H-indazole derivatives as novel selective bromodomain-containing protein 4 inhibitors. Bioorg Med Chem. 2021 Dec 29;55:116592. DOI:10.1016/j.bmc.2021.116592