Neladenoson dalanate (Neladenoson bialanate; BAY-1067197) hydrochloride is a orally active agonist precursor of partial Adenosine A1 Receptor. Neladenoson dalanate hydrochloride has a good pharmacokinetic and safety profile, can be used for the chronic heart diseases[1].
IC 50
A1R
References
[1] Meibom D, et al. Neladenoson Bialanate Hydrochloride: A Prodrug of a Partial Adenosine?A1 Receptor Agonist for the Chronic Treatment of Heart Diseases. ChemMedChem. 2017 May 22;12(10):728-737. DOI:10.1002/cmdc.201700151