S-(3-二甲氨基丙基)异硫脲二盐酸盐
S-(3-二甲氨基丙基)异硫脲二盐酸盐 性质
| 储存条件 | Desiccate at RT |
|---|---|
| 溶解度 | H2O：≥50mg/mL |
| 形态 | 粉末 |
| 颜色 | 白色至类白色 |
| 水溶解性 | Soluble to 100 mM in water |
S-(3-二甲氨基丙基)异硫脲二盐酸盐 用途与合成方法
|
H 2 Receptor
|
nNOS 49 μM (IC 50 ) |
Dimaprit has less than 0.0001% the activity of histamine on H1-receptors.
Dimaprit (0.1 nM-100 μM) inhibits nNOS concentration dependently with an IC
50
of 49±14 μM.
Dimaprit stimulates gastric acid secretion in rats (1.25 μM/kg/min; rapid i.v. injection), cats (2-64 μM/h; i.v.) and dogs (1-100 nM/kg/min; i.v.).
Dimaprit (0.01-1 μM/kg; i.v. at intervals of 5 min) causes dose-dependent falls in blood pressure in cats. Dimaprit (1-100 nM; intra-arterial injection) causes vasodilatation in the femoral vascular bed, and it (1 μM/kg; bolus or intravenous injection) has no effect on heart rate.
S-(3-二甲氨基丙基)异硫脲二盐酸盐 价格(试剂级)
| 更新日期 | 产品编号 | 产品名称 | CAS号 | 包装 | 价格 |
|---|---|---|---|---|---|
| 2024-04-30 | HY-B1478 | 25 mg | 600 | ||
| 2024-04-30 | HY-B1478 | 50 mg | 1000 |
