WAY-163909

WAY 163909 is a potent and selective 5-HT(2C) receptor agonist with a Ki of 10.5±1.1 nM.

5-HT_2C Receptor: 10.5±1.1 nM (Ki)

[1] Dunlop J,WAY-163909 [(7bR, 10aR)-1,2,3,4,8,9,10,10a-octahydro-7bH-cyclopenta-[b][1,4]diazepino[6,7,1hi]indole], a novel 5-hydroxytryptamine 2C receptor-selective agonist with anorectic activity. J Pharmacol Exp Ther. 2005 May; 313(2):862-9. Epub 2005 Feb 10. DOI:10.1124/jpet.104.075382