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托泊地芬

托泊地芬

中文名称:托泊地芬
英文名称:Tropodifene
CAS号:15790-02-0
分子式:C25H29NO4
分子量:407.507
EINECS号:
Mol文件:15790-02-0.mol
托泊地芬 结构式

托泊地芬 性质

沸点 508.5±50.0 °C(Predicted)
密度 1.20±0.1 g/cm3(Predicted)
储存条件 Store at -20°C
溶解度 溶于二甲基亚砜
酸度系数(pKa) 9.99±0.40(Predicted)

托泊地芬 用途与合成方法

Tropodifene (Tropaphen) 是α-肾上腺素能受体 (α-Adrenergic receptor) 抑制剂。

α-Adrenergic

Tropaphen has a beneficial effect on hypertension. The therapeutic effect of this preparation is more constant in diseases accompanied by spasm of the peripheral vessels. Tropaphen has a very marked adrenolytic and vasodilator action. It greatly lowers the tone of the peripheral vessels. The preparation is effective starting with a dose of 0.1 mg/kg. After injection of the drug in a dose of 0.25 mg/kg, a considerable and gradually progressive decrease in the perfusion pressure takes place. The pressure falls by 30-35% and remained at a low level for 90-100 min. With a dose of tropaphen of 0.5 mg/kg, the perfusion pressure falls by 40-45% and remains low for 120 min or more. Strong vasodilatation is also observed after injection of tropaphen into intact rabbits.

托泊地芬供应商 更多

天津普西唐生物医药科技有限公司
联系电话:010-60605840 15801484223
产品介绍:
中文名称:托泊地芬
英文名称:Tropodifene
CAS:15790-02-0
包装信息:100mg
备注: 试剂级
TargetMol中国(陶术生物)
联系电话: 4008200310
产品介绍:
中文名称:化合物 T13211
英文名称:Tropodifene;Tropodifene
CAS:15790-02-0
纯度:98%
包装信息:5 mg

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