DPP 728
中文名称:DPP 728
英文名称:DPP 728
CAS号:207556-62-5
分子式:C15H20Cl2N6O
分子量:371.2649
EINECS号:
Mol文件:207556-62-5.mol
![DPP 728 结构式](https://img.chemicalbook.com/CAS/20180906/GIF/207556-62-5.gif)
DPP 728 用途与合成方法
NVP-DPP728 dihydrochloride 是一种高效、选择性的二肽基肽酶 IV (DPP-IV) 抑制剂,其 Ki 为 11 nM。NVP-DPP728 dihydrochloride 可用于糖尿病的研究。
Ki: 11 nM (DPP-IV)
NVPDPP728 inhibits human and rat plasma DPP-IV (IC
50
s: 5-10 nM) with >15 000-fold selectivity relative to DPP-II and a range of proline-cleaving proteases.
NVP-DPP728 (3.72 mg/kg; p.o.) inhibits DPP-IV and improves insulin secretion and glucose tolerance, probably through augmentation of the effects of endogenous GLP-1.
Animal Model: | Obese (fa/fa) and lean (FA/?) Zucker rats |
Dosage: | 3.72 mg/kg |
Administration: | Oral administration |
Result: | Led to inhibition of plasma DPP-IV activity. |
DPP 728供应商 更多
天津普西唐生物医药科技有限公司
联系电话:010-60605840 15801484223;
产品介绍:
英文名称:NVP-DPP728 dihydrochloride
CAS:207556-62-5
包装信息:1mg
备注: 试剂级
銳迪國際科技有限公司
联系电话: 18024082417
产品介绍:
英文名称:NVP-DPP728 dihydrochloride
CAS:207556-62-5
纯度:5mg;10mg;50mg;100mg;250mg;500mg;1g
包装信息:5mg;10mg;50mg;100mg;250mg;500mg;1g