142479-62-7
142479-62-7 性质
| 沸点 | 969.3±65.0 °C(Predicted) |
|---|---|
| 密度 | 1.264±0.06 g/cm3(Predicted) |
| 储存条件 | −20°C |
| 溶解度 | 溶于二甲基亚砜 |
| 酸度系数(pKa) | 3.30±0.10(Predicted) |
| 形态 | 固体 |
| 颜色 | 白色至米白色 |
| 序列 | Tyr-Pro-Ile-Ser-Leu |
142479-62-7 用途与合成方法
IC50: 40 μM (μ opioid), 13.5 μM (δ opioid)
Gluten exorphin C, a novel opioid peptide, is isolated from the pepsin-trypsin-chymotrypsin digest of wheat gluten. Gluten exorphin C is evaluated its opioid activities by the GPI and MVD assays and its receptor affinities by radioreceptor assays. Its IC 50 s are 40 μM and 13.5 μM in the GPI and the MVD assays, respectively. Gluten exorphin C has a structure quite different from any of the endogenous and exogenous opioid peptides ever reported in that the N terminal Tyr is the only aromatic amino acid. The analogs containing Tyr-Pro-X-Ser-Leu are synthesized to study its structure-activity relationship. Peptides in which X is an aromatic amino acid or an aliphatic hydrophobic amino acid has opioid activity.
142479-62-7 价格(试剂级)
| 更新日期 | 产品编号 | 产品名称 | CAS号 | 包装 | 价格 |
|---|---|---|---|---|---|
| 2026-06-05 | HY-P1596 | 142479-62-7 | 142479-62-7 | 1 mg | 500 |
| 2026-06-05 | HY-P1596 | 142479-62-7 | 142479-62-7 | 5 mg | 1200 |