阻害剤活性化剤
- Chemical Name:WH-4-023 (SRC inhibitor)
- CAS:
- MF:
- Chemical Name:TG101348 (JAK inhibitor)
- CAS:
- MF:
- Chemical Name:PFI-3 (EPIGENETIC READER DOMAIN inhibitor)
- CAS:
- MF:
- Chemical Name:PD184352 (MEK inhibitor)
- CAS:
- MF:
- Chemical Name:ML324 (HISTONE DEMETHYLASE inhibitor)
- CAS:
- MF:
- Chemical Name:KU0063794 (MTOR inhibitor)
- CAS:
- MF:
- Chemical Name:JNJ-7777120 (HISTAMINE RECEPTOR antagonist)
- CAS:
- MF:
- Chemical Name:GSK1292263 (GPR agonist)
- CAS:
- MF:
- Chemical Name:BYL719 (PI3K inhibitor)
- CAS:
- MF:
- Chemical Name:BML-210 (HDAC inhibitor)
- CAS:
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- Structure:

- Chemical Name:2H-Pyran-4-propanamide, α-[4-(cyclopropylsulfonyl)phenyl]-N-(5-fluoro-2-thiazolyl)tetrahydro-, (αR)-
- CAS:745051-61-0
- MF:C20H23FN2O4S2
- Chemical Name:VENETOCLAX (ABT-199, GDC-0199) (BCL-2 inhibitor)
- CAS:
- MF:
- Chemical Name:U-104 (CARBONIC ANHYDRASE INHIBITOR)
- CAS:
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- Chemical Name:SALUBRINAL (PERK inhibitor)
- CAS:
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- Chemical Name:FLAVOPIRIDOL HCL (CDK inhibitor)
- CAS:
- MF:
- Chemical Name:DEFACTINIB (FAK inhibitor)
- CAS:
- MF:
- Chemical Name:CEDIRANIB (VEGFR inhibitor)
- CAS:
- MF:
- Chemical Name:BAY11-7082 (IΚB/IKK inhibitor)
- CAS:
- MF:
- Chemical Name:(-)-BLEBBISTATIN (ATPASE inhibitor)
- CAS:
- MF:
- Chemical Name:AG14361 (PARP1 inhibitor)
- CAS:
- MF:
- Chemical Name:ACP-196 (BTK inhibitor)
- CAS:
- MF:
- Chemical Name:ABT-737 (BCL-2 inhibitor)
- CAS:
- MF:
- Structure:

- Chemical Name:レルデセムチブ
- CAS:1345410-31-2
- MF:C19H18F2N6O
- Chemical Name:VILAZODONE (SSRI inhibitor)
- CAS:
- MF:
- Chemical Name:TBA-354 (anti-tuberculosis)
- CAS:
- MF:
- Chemical Name:SAG (HEDGEHOG/SMOOTHENED agonist)
- CAS:
- MF:
- Chemical Name:PACLITAXEL (MICROTUBULE ASSOSIATED inhibitor)
- CAS:
- MF:
- Chemical Name:OSU-03012 (PDK-1 inhibitor)
- CAS:
- MF:
- Chemical Name:MONOMETHYL AURISTATIN E (microtubule-associated inhibitor)
- CAS:
- MF:
- Chemical Name:ML141 (RHO inhibitor)
- CAS:
- MF:
- Chemical Name:KN-93 PHOSPHATE (CAMK Inhibitor)
- CAS:
- MF:
- Chemical Name:GSK126 (EZH2 inhibitor)
- CAS:
- MF:
- Chemical Name:GELDANAMYCIN (HSP90 inhibitor)
- CAS:
- MF:
- Chemical Name:GANT61 (HEDGEHOG/SMOOTHENED Inhibitor)
- CAS:
- MF:
- Chemical Name:EPZ-6438 (E7438) (EZH2 inhibitor)
- CAS:
- MF:
- Chemical Name:EMPAGLIFLOZIN (SGLT inhibitor)
- CAS:
- MF:
- Chemical Name:DOXORUBICIN (TOPOISOMERASE inhibitor)
- CAS:
- MF:
- Chemical Name:DAPT (Γ-SECRETASE inhibitor)
- CAS:
- MF:
- Chemical Name:DACLATASVIR (HCV NS5A inhibitor)
- CAS:
- MF:
- Chemical Name:COMBRETASTATIN A4 (MICROTUBULE ASSOCIATED inhibitor)
- CAS:
- MF:
- Chemical Name:CABOZANTINIB (VEGFR inhibitor)
- CAS:
- MF:
- Chemical Name:BREFELDIN A (protein transport inhibitor)
- CAS:
- MF:
- Chemical Name:BKM120 (PI3K inhibitor)
- CAS:
- MF:
- Chemical Name:AKT INHIBITOR VIII (AKT inhibitor)
- CAS:
- MF:
- Chemical Name:ABT-199 (BCL-2 inhibitor)
- CAS:
- MF:
- Chemical Name:VINCRISTINE (MICROTUBULE ASSOSIATED inhibitor)
- CAS:
- MF:
- Chemical Name:TETRABENAZINE (VMAT-2 Inhibitor)
- CAS:
- MF:
- Chemical Name:SNX-2112 (PF-04928473) (HSP90 antimony inhibitor)
- CAS:
- MF:
- Chemical Name:PLX4032 (RAF inhibitor)
- CAS:
- MF:
- Chemical Name:PD123319 (RAAS inhibitor)
- CAS:
- MF:
- Chemical Name:NS-2028 (SGC inhibitor)
- CAS:
- MF:
- Chemical Name:NECROSTATIN-1 (TNF-ALPHA inhibitor)
- CAS:
- MF:
- Chemical Name:ML323 (DUB inhibitor)
- CAS:
- MF:
- Chemical Name:KU-55933 (ATM inhibitor)
- CAS:
- MF:
- Chemical Name:(+)-JQ1 (BRD4 inhibitor)
- CAS:
- MF:
- Chemical Name:GSK2141795 (AKT inhibitor)
- CAS:
- MF:
- Chemical Name:GANETESPIB (HSP inhibitor)
- CAS:
- MF:
- Chemical Name:ENZALUTAMIDE (MDV3100) (AR inhibitor)
- CAS:
- MF:
- Chemical Name:BRIVANIB (VEGFR inhibitor)
- CAS:
- MF:
- Chemical Name:BARDOXOLONE METHYL (IΚB/IKK inhibitor)
- CAS:
- MF:
- Chemical Name:AZ20 (ATM/ATR inhibitor)
- CAS:
- MF:
- Chemical Name:ARN-509 (ANDROGEN RECEPTOR Inhibitor)
- CAS:
- MF:
- Structure:

- Chemical Name:3β-ヒドロキシ-20-オキソプレグナ-5-エン-16α-カルボニトリル
- CAS:1434-54-4
- MF:C22H31NO2
- Chemical Name:TWS119 (GSK-3 inhibitor)
- CAS:
- MF:
- Chemical Name:SC-514 (IΚB/IKK inhibitor)
- CAS:
- MF:
- Chemical Name:ROMIDEPSIN (HDAC inhibitor)
- CAS:
- MF:
- Chemical Name:REGADENOSON (ADENOSINE RECEPTOR agonist)
- CAS:
- MF:
- Chemical Name:PYRIDONE 6 (JAK inhibitor)
- CAS:
- MF:
- Chemical Name:PRT062607 HCL (SYK inhibitor)
- CAS:
- MF:
- Chemical Name:PAZOPANIB (VEGFR inhibitor)
- CAS:
- MF:
- Chemical Name:MLN9708 (20S PROTEASOME Inhibitor)
- CAS:
- MF:
- Chemical Name:INDIPLON (GABA RECEPTOR Conditioner)
- CAS:
- MF:
- Chemical Name:FIDAXOMICIN (DNA/RNA SYNTHESIS Inhibitor)
- CAS:
- MF:
- Chemical Name:EVEROLIMUS (MTOR inhibitor)
- CAS:
- MF:
- Chemical Name:ENTOSPLETINIB (SYK inhibitor)
- CAS:
- MF:
- Chemical Name:DABRAFENIB (RAF inhibitor)
- CAS:
- MF:
- Chemical Name:CYT997 (LEXIBULIN) (MICROTUBULES inhibitor)
- CAS:
- MF:
- Chemical Name:BMS-5 (LIMK inhibitor)
- CAS:
- MF:
- Chemical Name:AZD7762 (CHK inhibitor)
- CAS:
- MF:
- Chemical Name:AG1024 (IGF-1R inhibitor)
- CAS:
- MF:
- Chemical Name:VISMODEGIB (HEDGEHOG/SMOOTHENED INHIBITOR)
- CAS:
- MF:
- Chemical Name:REMODELIN (HISTONE ACETYLTRANSFERASE inhibitor)
- CAS:
- MF:
- Chemical Name:PAC-1 (CASPASE Activator)
- CAS:
- MF:
- Chemical Name:OSELTAMIVIR PHOSPHATE (NEURAMINIDASE Inhibitor)
- CAS:
- MF:
- Chemical Name:MONENSIN (protein transport inhibitor)
- CAS:
- MF:
- Chemical Name:LINIFANIB (VEGFR inhibitor)
- CAS:
- MF:
- Chemical Name:LCZ696 (RAAS inhibitor)
- CAS:
- MF:
- Chemical Name:IONOMYCIN (calcium ionophore)
- CAS:
- MF:
- Chemical Name:HYDROXYUREA (DNA SYNTHESIS inhibitor)
- CAS:
- MF:
- Chemical Name:GZD824 DIMESYLATE (BCR-ABL inhibitor)
- CAS:
- MF:
- Chemical Name:FORETINIB (C-MET inhibitor)
- CAS:
- MF:
- Chemical Name:DAPIVIRINE (REVERSE TRANSCRIPTASE Inhibitor)
- CAS:
- MF:
- Chemical Name:CNX-774 (BTK inhibitor)
- CAS:
- MF:
- Chemical Name:BIRB 796 (P38 MAPK Inhibitor)
- CAS:
- MF:
- Chemical Name:BAY87-2243 (HIF inhibitor)
- CAS:
- MF:
- Chemical Name:B-AP15 (DUB inhibitor)
- CAS:
- MF:
- Chemical Name:APIXABAN (FACTOR XA Inhibitor)
- CAS:
- MF:
- Chemical Name:TPA Deficient Plasma
- CAS:
- MF:

